SCHEMBL16712945

SCHEMBL16712945

COc1cccc(-c2cc(C(C)C)ccc2O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPN5 P54829 1/20 0.52
AKR1C3 P42330 3/20 0.50
AKR1C2 P52895 3/20 0.50
HDAC4 P56524 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
AKR1C4 P17516 1/20 0.47
AKR1C1 Q04828 1/20 0.47
RXRA P19793 1/20 0.47
NR4A2 P43354 1/20 0.47
THRA P10827 2/20 0.46
THRB P10828 2/20 0.46
FYN P06241 1/20 0.44
GPR35 Q9HC97 1/20 0.43
HDAC2 Q92769 1/20 0.43
TRPA1 O75762 1/20 0.42
PTGS1 P23219 1/20 0.42
CACNA1C Q13936 1/20 0.42
SERPINE1 P05121 1/20 0.42
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16710322 0.84 LMNA (0.50) AKR1C3AKR1C2AKR1C4AKR1C1TRPA1
SCHEMBL6934499 0.83 HDAC4 (0.50) AKR1C3AKR1C2HDAC4HDAC8AKR1C4
SCHEMBL26378188 0.82 AKR1C3 (0.56) AKR1C3AKR1C2AKR1C4AKR1C1CYP1A1
SCHEMBL27632212 0.81 MIF (0.55) HDAC4HDAC8THRATHRBFYN
SCHEMBL18087561 0.80 ACHE (0.53) HDAC4HDAC8THRATHRBFYN
SCHEMBL18084773 0.80 PTPN5 (0.56) PTPN5AKR1C3AKR1C2HDAC4HDAC8
SCHEMBL487170 0.79 CYP1A1 (0.53) AKR1C3AKR1C2HDAC4HDAC8RXRA
SCHEMBL4282140 0.79 PTPN5 (0.57) PTPN5AKR1C3AKR1C2HDAC4HDAC8
SCHEMBL6572257 0.78 FYN (0.55) HDAC4HDAC8THRATHRBFYN
SCHEMBL16429142 0.78 HDAC4 (0.51) AKR1C3AKR1C2HDAC4HDAC8THRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3066072-B1 BIPHENYLAMIDE DERIVATIVE HSP90 INHIBITORS UNIV KANSAS (US) 2021-11-03 EP disclosed
WO-2015070091-A1 BIPHENYLAMIDE DERIVATIVE HSP90 INHIBITORS THE UNIVERSITY OF KANSAS (US) 2015-05-14 WO disclosed