SCHEMBL16719476

SCHEMBL16719476

Oc1cccc(-c2nc[c]cn2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 13/20 0.61
HSD17B2 P37059 13/20 0.61
CYP3A4 P08684 4/20 0.50
CYP2C9 P11712 3/20 0.50
CYP19A1 P11511 1/20 0.45
METAP2 P50579 1/20 0.44
ESR1 P03372 2/20 0.42
ESR2 Q92731 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2B6 P20813 1/20 0.42
CYP2C19 P33261 1/20 0.42
CA12 O43570 1/20 0.42
ALDH1A1 P00352 1/20 0.42
CA2 P00918 1/20 0.42
LMNA P02545 1/20 0.42
CA5A P35218 1/20 0.42
CA9 Q16790 1/20 0.42
HSD17B10 Q99714 1/20 0.42
CA14 Q9ULX7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27625438 0.81 HSD17B1 (0.68) HSD17B1HSD17B2CYP3A4CYP2C9CYP19A1
SCHEMBL27905669 0.78 HSD17B1 (0.63) HSD17B1HSD17B2CYP3A4CYP2C9CYP19A1
SCHEMBL29444135 0.76 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2C9CYP19A1
SCHEMBL23868941 0.76 HSD17B1 (0.74) HSD17B1HSD17B2CYP3A4CYP2C9CYP19A1
SCHEMBL1180643 0.76 HSD17B1 (1.00) HSD17B1HSD17B2CYP3A4CYP2C9CYP19A1
SCHEMBL16719539 0.76 HPGDS (0.47) ESR2
SCHEMBL27813877 0.76 PRKCI (0.51) PIK3CDPIK3CA
SCHEMBL4775356 0.76 HSD17B1 (0.56) HSD17B1HSD17B2CYP3A4CYP2C9CYP19A1
SCHEMBL21944933 0.74 HSD17B1 (0.59) HSD17B1HSD17B2CYP3A4CYP2C9CYP19A1
SCHEMBL27612450 0.74 NPC1 (0.63) HSD17B1HSD17B2CYP3A4CYP2C9METAP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed