SCHEMBL16719495

SCHEMBL16719495

[c]1ccc2[nH]c(-c3ccncc3)nc2c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.60
PKN1 Q16512 4/20 0.60
PKN2 Q16513 4/20 0.60
KDM4E B2RXH2 4/20 0.60
HPGD P15428 4/20 0.51
HSD17B10 Q99714 2/20 0.51
RHEB Q15382 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
CYP2C19 P33261 1/20 0.51
NPC1 O15118 4/20 0.50
RAB9A P51151 3/20 0.50
GAA P10253 3/20 0.43
PKM P14618 2/20 0.43
MGAM O43451 1/20 0.43
SI P14410 1/20 0.43
MGAM2 Q2M2H8 1/20 0.43
MAPT P10636 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316190 0.87 ALDH1A1 (0.60) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL694906 0.85 NPC1 (0.62) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL9033788 0.82 NPC1 (0.53) ALDH1A1KDM4EHPGDHSD17B10RHEB
SCHEMBL695765 0.82 KDM4E (0.61) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL704211 0.81 NPBWR1 (0.51)
SCHEMBL2124653 0.81 KDM4E (0.66) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL5543777 0.80 KDM4E (0.37) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL2079577 0.80 RHEB (0.57) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL2078169 0.79 KDM4E (0.38) ALDH1A1PKN1PKN2KDM4EHPGD
SCHEMBL9032674 0.77 KDM4E (0.63) ALDH1A1KDM4EHPGDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed