SCHEMBL16719829

SCHEMBL16719829

[c]1nccc(-c2ccc3cc[nH]c3c2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.42
APP P05067 1/20 0.42
NISCH Q9Y2I1 1/20 0.41
AHR P35869 3/20 0.41
CMA1 P23946 1/20 0.41
TYR P14679 1/20 0.41
BRAF P15056 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
CCNC P24863 1/20 0.38
CDK8 P49336 1/20 0.38
ENPP2 Q13822 2/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP2A6 P11509 1/20 0.38
DYRK1B Q9Y463 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654046 0.75 CYP1A2 (0.47) NISCHMEN1KMT2AKDM4EALDH1A1
SCHEMBL29445919 0.72 BRAF (0.47) BRD4APPAHRCMA1TYR
SCHEMBL4786964 0.71 AHR (0.49) BRD4APPNISCHAHRCMA1
SCHEMBL18000228 0.70 BRAF (0.58) BRD4AHRCMA1TYRBRAF
SCHEMBL6460701 0.70 NISCH (0.53) BRD4NISCHMEN1KMT2ADYRK1B
SCHEMBL16719949 0.70 ADORA2A (0.42) BRD4APPNISCHAHRCMA1
SCHEMBL16720139 0.70 ADORA2A (0.42) BRD4APPNISCHAHRCMA1
SCHEMBL17626014 0.69 KMO (0.49) AHRMEN1KMT2AKDM4EALDH1A1
SCHEMBL18828549 0.69 BACE1 (0.47) BRD4APPAHRCMA1TYR
SCHEMBL27361728 0.69 BRD4 (0.46) BRD4APPAHRCMA1TYR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed