SCHEMBL4786964

SCHEMBL4786964

Clc1nccc(-c2ccc3cc[nH]c3c2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 3/20 0.49
CMA1 P23946 1/20 0.49
BRAF P15056 1/20 0.43
BRD4 O60885 1/20 0.42
APP P05067 1/20 0.42
KDM4C Q9H3R0 1/20 0.41
CHRNA7 P36544 2/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA10 Q9GZZ6 1/20 0.41
CHRNA9 Q9UGM1 1/20 0.41
KMO O15229 2/20 0.41
TYR P14679 1/20 0.41
KCNH2 Q12809 2/20 0.40
MPO P05164 1/20 0.40
TPO P07202 1/20 0.40
DYRK1B Q9Y463 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
SYK P43405 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3400660 0.87 AHR (0.49) AHRBRAFBRD4APPKMO
SCHEMBL9213361 0.77 MAPT (0.51) BRD4APPKDM4CADORA2AADORA1
SCHEMBL29445919 0.75 BRAF (0.47) AHRCMA1BRAFBRD4APP
SCHEMBL19133030 0.75 MAP4K4 (0.47) KMOKCNH2
SCHEMBL445861 0.75 MEN1 (0.52) KMO
SCHEMBL27084041 0.74 CCR1 (0.50) AHRCMA1BRAFBRD4KDM4C
SCHEMBL7544652 0.74 KMO (0.69) AHRKMODYRK1B
SCHEMBL12520573 0.73 SYK (0.47) AHRCMA1APPSYKAURKA
SCHEMBL27361728 0.73 BRD4 (0.46) AHRCMA1BRAFBRD4APP
SCHEMBL18828549 0.73 BACE1 (0.47) AHRCMA1BRAFBRD4APP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008060248-A1 INDOLE SUSTITUTED PYRIMIDINES AND USE THEREOF IN THE TREATMENT OF CANCER S*BIO PTE LTD. (SG) 2008-05-22 WO disclosed
WO-2008060248-A1 INDOLE SUSTITUTED PYRIMIDINES AND USE THEREOF IN THE TREATMENT OF CANCER S*BIO PTE LTD. (SG) 2008-05-22 WO disclosed