SCHEMBL16719901

SCHEMBL16719901

COc1cc(O)cc(-c2cc[c]cc2O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 5/20 0.44
ABCB1 P08183 5/20 0.44
BCR P11274 5/20 0.44
TP53 P04637 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
MAPK1 P28482 1/20 0.42
CASP3 P42574 1/20 0.42
RAB9A P51151 1/20 0.42
SENP8 Q96LD8 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
CYP3A4 P08684 2/20 0.39
TTR P02766 1/20 0.38
CYP1A1 P04798 1/20 0.38
ALOX5 P09917 1/20 0.38
PTGS2 P35354 1/20 0.38
CYP1B1 Q16678 1/20 0.38
CALM1 P0DP23 2/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16719990 0.85 ABL1 (0.39) ABL1ABCB1BCRNPC1RAB9A
SCHEMBL2377419 0.81 HDAC4 (0.50) ABL1ABCB1BCRCYP3A4CYP1A1
SCHEMBL16719656 0.80 ESR2 (0.47) ABL1ABCB1BCRTP53SMN1; SMN2
SCHEMBL16720630 0.79 CYP11B1 (0.47) CYP3A4CYP1A1CYP1B1
SCHEMBL16719854 0.78 ABL1 (0.34) ABL1ABCB1BCRTP53SMN1; SMN2
SCHEMBL16719523 0.76 HSD17B1 (0.40) ABL1ABCB1BCRESR2
SCHEMBL16720192 0.76 CNR1 (0.39) ABL1ABCB1BCRALOX5
SCHEMBL17514940 0.72 AKR1C3 (0.44) ABL1ABCB1BCRCYP3A4CYP1A1
SCHEMBL17514647 0.72 ABL1 (0.43) ABL1ABCB1BCRCYP3A4CYP1A1
SCHEMBL2850768 0.71 KMT2A (0.49) TP53SMN1; SMN2NPC1MAPK1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed