SCHEMBL16720131

SCHEMBL16720131

Oc1ccc[c]c1-c1cccc(F)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.47
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41
MAPT P10636 2/20 0.40
ALOX15 P16050 2/20 0.40
NFKB1 P19838 2/20 0.40
NFKB2 Q00653 2/20 0.40
RELA Q04206 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 1/20 0.40
ALOX12 P18054 1/20 0.40
MAPK1 P28482 1/20 0.40
TAAR1 Q96RJ0 3/20 0.39
NQO2 P16083 1/20 0.39
PTGS1 P23219 1/20 0.39
APP P05067 1/20 0.35
NOTUM Q6P988 2/20 0.35
NR4A1 P22736 1/20 0.35
NR4A2 P43354 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10494072 0.81 TAAR1 (0.41) ESR2HSD17B1HSD17B2MAPTTAAR1
SCHEMBL9987901 0.81 HSD17B1 (0.48) ESR2HSD17B1HSD17B2LMNA
SCHEMBL16719521 0.81 HSD17B1 (0.40) ESR2HSD17B1HSD17B2MAPTALOX15
SCHEMBL9650164 0.79 NPC1 (0.35) HSD17B1HSD17B2MAPTALOX15NFKB1
SCHEMBL16720373 0.79 ACHE (0.41) RAB9A
SCHEMBL2012944 0.79 MGAM (0.42) ESR2HSD17B1HSD17B2TAAR1NOTUM
SCHEMBL2013348 0.79 TAAR1 (0.39) ESR2HSD17B1HSD17B2TAAR1NOTUM
SCHEMBL16719910 0.79 ALOX5 (0.55) ESR2ALOX15NFKB1NFKB2RELA
SCHEMBL16719822 0.79 HSD17B1 (0.47) ESR2HSD17B1HSD17B2LMNA
SCHEMBL16720445 0.78 ESR2 (0.40) ESR2HSD17B1HSD17B2SMN1; SMN2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3068758-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE The Wistar Institute Of Anatomy And Biology (US) 2016-09-21 EP disclosed
WO-2015073864-A1 EBNA1 INHIBITORS AND THEIR METHOD OF USE THE WISAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2015-05-21 WO disclosed