SCHEMBL1672246

SCHEMBL1672246

Cc1ccc2c(c(CNC3CN4CCC3CC4)nn2C(C)C)c1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
HTR3A P46098 3/20 0.36
CHRNA7 P36544 2/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
TSHR P16473 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1672705 0.91 SIGMAR1 (0.37) HTR3ACHRNA7ALDH1A1CYP1A2CYP3A4
SCHEMBL1673270 0.87 GAA (0.38) GAASMN1; SMN2MEN1KMT2ACHRNA7
SCHEMBL1672396 0.87 GAA (0.35) GAASMN1; SMN2MEN1KMT2AHTR3A
SCHEMBL1672241 0.86 GAA (0.37) GAASMN1; SMN2MEN1KMT2AHTR3A
SCHEMBL701669 0.84 HTR3A (0.42) GAAHTR3A
SCHEMBL4311850 0.84 HTR3A (0.42) GAAHTR3A
SCHEMBL701670 0.84 HTR3A (0.42) GAAHTR3A
SCHEMBL700430 0.83 HTR3A (0.42) GAAHTR3ACYP1A2CYP2C9
SCHEMBL1672707 0.82 MEN1 (0.47) GAASMN1; SMN2MEN1KMT2ACHRNA7
SCHEMBL1673275 0.79 GAA (0.32) GAASMN1; SMN2MEN1KMT2AHTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2310019-A2 5-HT3 RECEPTOR MODULATORS, METHODS OF MAKING, AND USE THEREOF Albany Molecular Research, Inc. (US) 2011-04-20 EP disclosed
WO-2009155054-A2 5-HT3 RECEPTOR MODULATORS, METHODS OF MAKING, AND USE THEREOF ALBANY MOLECULAR RESEARCH, INC. (US) 2009-12-23 WO disclosed