SCHEMBL1672807

SCHEMBL1672807

Cc1noc(C)c1-c1c(-c2ccc(O)cc2)cn(C)c1C(N)=NO

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 14/20 0.38
BRD2 P25440 1/20 0.37
MLYCD O95822 1/20 0.36
ERN1 O75460 1/20 0.34
HSP90AB1 P08238 1/20 0.34
CREBBP Q92793 3/20 0.33
USP7 Q93009 1/20 0.33
BRAF P15056 1/20 0.32
MAPK3 P27361 1/20 0.32
MAPK1 P28482 1/20 0.32
AR P10275 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1672805 1.00 BRD4 (0.38) BRD4BRD2MLYCDERN1HSP90AB1
SCHEMBL1672861 0.91 BRD4 (0.38) BRD4BRD2MLYCDERN1CREBBP
SCHEMBL1672863 0.91 BRD4 (0.38) BRD4BRD2MLYCDERN1CREBBP
SCHEMBL12800384 0.86 BRD4 (0.39) BRD4BRD2MLYCDERN1HSP90AB1
SCHEMBL1672789 0.85 ERN1 (0.38) BRD4BRD2MLYCDERN1
SCHEMBL1672787 0.85 ERN1 (0.38) BRD4BRD2MLYCDERN1
SCHEMBL1670718 0.84 TLR8 (0.41) BRD4BRD2MLYCDCREBBP
SCHEMBL1670714 0.84 TLR8 (0.41) BRD4BRD2MLYCDCREBBP
SCHEMBL1670492 0.84 BRD4 (0.35) BRD4ERN1HSP90AB1CREBBPAR
SCHEMBL1670734 0.81 MLYCD (0.38) BRD4BRD2MLYCDERN1CREBBP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011042477-A1 SUBSTITUTED PYRROLES AND IMIDAZOLES AS ESTROGEN RECEPTOR LIGANDS KARO BIO AB (SE) 2011-04-14 WO disclosed