SCHEMBL1673073

SCHEMBL1673073

Cc1ccc2c(c(CCNC3CN4CCC3CC4)cn2C)c1C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.40
CHRM1 P11229 3/20 0.40
CHRM3 P20309 3/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
HTR2A P28223 2/20 0.40
HTR2C P28335 2/20 0.40
HTR4 Q13639 2/20 0.40
CYP1A2 P05177 1/20 0.40
CHRM4 P08173 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
HTR1D P28221 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
SIGMAR1 Q99720 1/20 0.40
CHRNA7 P36544 3/20 0.35
CDK2 P24941 1/20 0.35
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1672238 0.84 HTR6 (0.41) HTR1DSIGMAR1CHRNA7
SCHEMBL4324945 0.83 CHRM2 (0.48) CHRM2CHRM1CHRM3ADRA2AADRA2B
SCHEMBL4324940 0.83 CHRM2 (0.48) CHRM2CHRM1CHRM3ADRA2AADRA2B
SCHEMBL4325921 0.83 CHRM2 (0.48) CHRM2CHRM1CHRM3ADRA2AADRA2B
SCHEMBL700017 0.82 CHRM2 (0.47) CHRM2CHRM1CHRM3ADRA2AADRA2B
SCHEMBL1672448 0.82 SIGMAR1 (0.39) CHRM2CHRM1CHRM3ADRA2AADRA2B
SCHEMBL1672243 0.78 SIGMAR1 (0.38) SIGMAR1CHRNA7
SCHEMBL702139 0.78 CHRM2 (0.48) CHRM2CHRM1CHRM3ADRA2AADRA2B
SCHEMBL702645 0.78 CHRM2 (0.48) CHRM2CHRM1CHRM3ADRA2AADRA2B
Lithium Ion SCHEMBL703148 0.78 CHRM2 (0.46) CHRM2CHRM1CHRM3ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2310019-A2 5-HT3 RECEPTOR MODULATORS, METHODS OF MAKING, AND USE THEREOF Albany Molecular Research, Inc. (US) 2011-04-20 EP disclosed
WO-2009155054-A2 5-HT3 RECEPTOR MODULATORS, METHODS OF MAKING, AND USE THEREOF ALBANY MOLECULAR RESEARCH, INC. (US) 2009-12-23 WO disclosed