SCHEMBL16740643

SCHEMBL16740643

Oc1ccc(C2CC(c3ccccc3O)=NN2c2ccc(Cl)cc2)cc1O

nearest known ligand 0.78

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PRKCZ Q05513 12/20 0.78
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
HSP90AA1 P07900 1/20 0.63
ATM Q13315 1/20 0.63
ESD P10768 1/20 0.53
PDE5A O76074 1/20 0.53
EGFR P00533 1/20 0.52
ERBB2 P04626 1/20 0.52
MAOA P21397 2/20 0.52
MAOB P27338 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16740593 0.88 PRKCZ (1.00) PRKCZMEN1KMT2AHSP90AA1ATM
SCHEMBL16740631 0.79 PRKCZ (1.00) PRKCZMEN1KMT2AHSP90AA1ATM
SCHEMBL16740663 0.78 PRKCZ (1.00) PRKCZMEN1KMT2AHSP90AA1ATM
SCHEMBL27792765 0.76 PRKCZ (0.67) PRKCZMEN1KMT2AHSP90AA1ATM
SCHEMBL16740616 0.74 PRKCZ (0.73) PRKCZMEN1KMT2AHSP90AA1PDE5A
SCHEMBL16740622 0.74 CA1 (0.63) PRKCZMEN1KMT2AATMPDE5A
SCHEMBL16740611 0.73 PRKCZ (1.00) PRKCZMEN1KMT2AHSP90AA1ATM
SCHEMBL9628590 0.73 PRKCZ (1.00) PRKCZMEN1KMT2AHSP90AA1ATM
SCHEMBL16740614 0.71 PRKCZ (0.69) PRKCZMEN1KMT2AHSP90AA1ATM
SCHEMBL16740640 0.70 PRKCZ (1.00) PRKCZMEN1KMT2AHSP90AA1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230192904-A1 BIFUNCTIONAL CHIMERIC MOLECULES FOR LABELING OF KINASES WITH TARGET BINDING MOIETIES AND METHODS OF USE THEREOF THE BROAD INSTITUTE, INC. 2023-06-22 US disclosed
US-20230192904-A1 BIFUNCTIONAL CHIMERIC MOLECULES FOR LABELING OF KINASES WITH TARGET BINDING MOIETIES AND METHODS OF USE THEREOF THE BROAD INSTITUTE, INC. 2023-06-22 US disclosed
WO-2015075051-A1 ALLOSTERIC INHIBITORS OF ATYPICAL PROTEIN KINASES C UNIVERSITAET DES SAARLANDES (DE) 2015-05-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230192904-A1 BIFUNCTIONAL CHIMERIC MOLECULES FOR LABELING OF KINASES WITH TARGET BINDING MOIETIES AND METHODS OF USE THEREOF ERBB2, ACP1, TK1 PRKCZ 25/4885MEN1 3627/4885KMT2A 1636/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.