SCHEMBL16757264

SCHEMBL16757264

COC(=O)[C@@H]1CCN2C(CO[Si](C)(C)C(C)(C)C)CCC12

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.30
FKBP1A P62942 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16757219 0.77 CYP1A2 (0.34) SMN1; SMN2
SCHEMBL16760697 0.76 TDP1 (0.31)
SCHEMBL29132569 0.74 FKBP1A (0.32) FKBP1A
SCHEMBL17961794 0.72 SMN1; SMN2 (0.34) SMN1; SMN2FKBP1A
SCHEMBL17961792 0.72 SMN1; SMN2 (0.34) SMN1; SMN2FKBP1A
SCHEMBL16579348 0.72 SMN1; SMN2 (0.34) SMN1; SMN2FKBP1A
SCHEMBL16579389 0.72 SMN1; SMN2 (0.34) SMN1; SMN2FKBP1A
SCHEMBL31153913 0.69 RECQL (0.38) SMN1; SMN2
SCHEMBL29132593 0.68 SMN1; SMN2 (0.41) SMN1; SMN2FKBP1A
SCHEMBL27089375 0.68

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3074402-A1 BICYCLOAMINE-SUBSTITUTED-N-BENZENESULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS Merck Sharp & Dohme Corp. (US) 2016-10-05 EP disclosed
WO-2015077905-A1 BICYCLOAMINE-SUBSTITUTED-N-BENZENESULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS MERCK SHARP & DOHME CORP. (US) 2015-06-04 WO disclosed
WO-2015080988-A1 BICYCLOAMINE-SUBSTITUTED-N-BENZENESULFONAMIDE COMPOUNDS WITH SELECTIVE ACTIVITY IN VOLTAGE-GATED SODIUM CHANNELS MERCK SHARP & DOHME CORP. (US) 2015-06-04 WO disclosed