SCHEMBL16759793

SCHEMBL16759793

FC(F)F.O=C(O)c1ccc2cc[nH]c2c1

nearest known ligand 0.86

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.86
HSD17B10 Q99714 2/20 0.86
KDM4E B2RXH2 2/20 0.86
ENPP2 Q13822 2/20 0.86
HPGD P15428 1/20 0.86
GHSR Q92847 2/20 0.50
TAS1R3 Q7RTX0 1/20 0.50
TAS1R1 Q7RTX1 1/20 0.50
ESR1 P03372 3/20 0.49
TYR P14679 1/20 0.47
AHR P35869 1/20 0.47
MAPT P10636 2/20 0.47
MAPK14 Q16539 2/20 0.46
CHRNA7 P36544 1/20 0.46
SMYD3 Q9H7B4 1/20 0.45
HDAC3 O15379 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL50542 0.93 ALDH1A1 (1.00) ALDH1A1HSD17B10KDM4EENPP2HPGD
SCHEMBL4595294 0.93 ALDH1A1 (1.00) ALDH1A1HSD17B10KDM4EENPP2HPGD
SCHEMBL29583385 0.93 ALDH1A1 (1.00) ALDH1A1HSD17B10KDM4EENPP2HPGD
Hydrochloric Acid SCHEMBL1373044 0.91 ALDH1A1 (0.96) ALDH1A1HSD17B10KDM4EENPP2HPGD
Hydrazine SCHEMBL27365039 0.89 ALDH1A1 (0.93) ALDH1A1HSD17B10KDM4EENPP2HPGD
Trifluoroacetic Acid SCHEMBL5740837 0.87 ALDH1A1 (0.81) ALDH1A1HSD17B10KDM4EENPP2HPGD
Indole SCHEMBL28009908 0.80 ALDH1A1 (0.73) ALDH1A1HSD17B10KDM4EENPP2HPGD
SCHEMBL2951840 0.79 KDM4E (0.74) ALDH1A1HSD17B10KDM4EENPP2HPGD
SCHEMBL105928 0.78 KDM4E (0.72) ALDH1A1HSD17B10KDM4EENPP2HPGD
Benzoic Acid SCHEMBL8915824 0.78 ALDH1A1 (0.71) ALDH1A1HSD17B10KDM4EENPP2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3074400-A1 NEW OCTAHYDRO-CYCLOBUTA [1,2-c;3,4-c']DIPYRROL-2-YL F. Hoffmann-La Roche AG (CH) 2016-10-05 EP disclosed
WO-2015078803-A1 NEW OCTAHYDRO-CYCLOBUTA [1,2-c;3,4-c']DIPYRROL-2-YL F. HOFFMANN-LA ROCHE AG (CH) 2015-06-04 WO disclosed