SCHEMBL16772146

SCHEMBL16772146

N#CC(C#N)=C1C=CC(=O)C(c2ccc(C(F)(F)F)cc2C(F)(F)F)=C1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.37
AR P10275 5/20 0.34
EDNRB P24530 1/20 0.33
EDNRA P25101 1/20 0.33
POLQ O75417 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
ALDH1A1 P00352 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
TDP2 O95551 1/20 0.30
FLT1 P17948 1/20 0.30
FLT4 P35916 1/20 0.30
KDR P35968 1/20 0.30
BACE1 P56817 1/20 0.30
TMPRSS4 Q9NRS4 1/20 0.30
ESRRA P11474 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16772037 0.81 BACE1 (0.49) CES2BACE1
SCHEMBL16769520 0.79 PTPN11 (0.42) CES2EDNRBEDNRAABCC8KCNJ11
SCHEMBL16772055 0.73 CES2 (0.42) CES2AREDNRBEDNRAPOLQ
SCHEMBL10075607 0.68 EDNRB (0.42) CES2AREDNRBEDNRAPOLQ
SCHEMBL16772093 0.67
SCHEMBL28676412 0.66 TSHR (0.56) CES2AREDNRBEDNRAABCC8
SCHEMBL13302009 0.65 MAPT (0.45) CES2ALDH1A1TDP2
SCHEMBL11588370 0.65 HPRT1 (0.39) CES2ARPOLQALDH1A1ESRRA
SCHEMBL16772040 0.64 CES2 (0.42) CES2ARPOLQALDH1A1HTT
SCHEMBL24397228 0.64 TDP2 (0.40) CES2TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150155490-A1 ORGANIC COMPOUNDS AND ORGANIC LIGHT EMITTING DEVICE COMPRISING THE SAME LG DISPLAY CO., LTD. (KR) 2015-06-04 US disclosed