SCHEMBL16775445

SCHEMBL16775445

COC(=O)c1ccc(-n2ccc(-c3ccc(C(=O)O)cc3)c2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.54
ADH5 P11766 1/20 0.51
ALDH1A1 P00352 5/20 0.45
ALDH1A3 P47895 1/20 0.45
PTPN1 P18031 1/20 0.43
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA9 Q16790 2/20 0.43
CA14 Q9ULX7 2/20 0.43
KDM4E B2RXH2 1/20 0.43
PKM P14618 1/20 0.43
HPGD P15428 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
EGFR P00533 1/20 0.43
TSHR P16473 1/20 0.42
RXRA P19793 1/20 0.42
SETD7 Q8WTS6 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CA7 P43166 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10195813 0.88 ADH5 (0.63) ADH5TSHRRXRA
SCHEMBL182048 0.86 CA1 (0.57) ADH5ALDH1A1CA1CA2KDM4E
SCHEMBL182128 0.84 HTT (0.49) HTTALDH1A1PTPN1CA12CA1
SCHEMBL182280 0.84 ADH5 (0.55) HTTADH5ALDH1A1CA12CA1
SCHEMBL181958 0.83 ALDH1A1 (0.57) ADH5ALDH1A1KDM4ERXRAMEN1
SCHEMBL182263 0.82 ADH5 (0.55) ADH5EGFRTSHR
SCHEMBL204640 0.81 TSHR (0.61) ALDH1A1PTPN1CA12CA1CA2
SCHEMBL2710630 0.81 BCL2L1 (0.62) ADH5KDM4ERXRAMEN1KMT2A
SCHEMBL182188 0.81 ADH5 (0.55) ADH5ALDH1A1KDM4ETSHRRXRA
SCHEMBL181985 0.80 ADH5 (0.51) ADH5ALDH1A1HPGDRXRAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9051342-B2 Pyrazole or triazole compounds and their use for the manufacture of a medicament for treating somatic mutation related diseases PTC THERAPEUTICS, INC. (US) 2015-06-09 US disclosed