SCHEMBL16795802

SCHEMBL16795802

C=C(CO)c1cccc(-c2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.52
PRSS1 P07477 1/20 0.50
PRSS2 P07478 1/20 0.50
PRSS3 P35030 1/20 0.50
ERCC5 P28715 1/20 0.47
FEN1 P39748 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
NR1H4 Q96RI1 2/20 0.41
GPR52 Q9Y2T5 1/20 0.41
EPHX2 P34913 1/20 0.41
DHODH Q02127 1/20 0.40
MGLL Q99685 1/20 0.39
GRIK2 Q13002 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10204736 0.81 SMN1; SMN2 (0.45) ERCC5FEN1
SCHEMBL38664634 0.81 KMO (0.48) KMOPRSS1PRSS2PRSS3ERCC5
SCHEMBL93850 0.80 MAOA (0.54)
SCHEMBL13442275 0.79 KMO (0.59) KMOPRSS1PRSS2PRSS3ERCC5
SCHEMBL16795663 0.77 PRSS1 (0.56) PRSS1PRSS2PRSS3
SCHEMBL2070299 0.76 ERCC5 (0.66) KMOPRSS1PRSS2PRSS3ERCC5
SCHEMBL20243662 0.75 PRSS1 (0.64) KMOPRSS1PRSS2PRSS3ERCC5
SCHEMBL2135450 0.75 KMO (0.55) KMOPRSS1PRSS2PRSS3ERCC5
SCHEMBL26828809 0.74 PRSS1 (0.49) KMOPRSS1PRSS2PRSS3ERCC5
SCHEMBL28604413 0.73 PARP1 (0.48) ERCC5FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015087094-A1 NEW ARYLALKENYLPROPARGYLAMINE DERIVATIVES EXHIBITING NEUROPROTECTIVE ACTION FOR THE TREATMENT OF NEURODEGENERATIVE DISEASES SEMMELWEIS EGYETEM (HU) 2015-06-18 WO disclosed
CN-1040321-C Pyran-2-ones and 5,6-dihydropyran-2-ones useful for treating HIV and other retroviruses UPJOHN CO (US) 1998-10-21 CN disclosed
CN-1090279-A Be used for the treatment of HIV and other retroviral pyran-2-ones and 5,6-dihydropyrane-2-ketone UPJOHN CO (US) 1994-08-03 CN disclosed