SCHEMBL16799547

SCHEMBL16799547

CC1(c2ccc(Br)cc2)CCc2nc(Cl)ccc2C1=O

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.36
HTR6 P50406 1/20 0.32
HSD17B10 Q99714 1/20 0.31
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16798942 0.89 GRM5 (0.37) GRM5HTR6HSD11B1
SCHEMBL16800949 0.87 GRM5 (0.36) GRM5HTR6HSD11B1
SCHEMBL16801068 0.86 GRM5 (0.45) GRM5HSD11B1
SCHEMBL16798949 0.85 GRM5 (0.34) GRM5HTR6HSD17B10
SCHEMBL16800681 0.85 MAPT (0.38) GRM5HTR6HSD17B10
SCHEMBL16799448 0.84 CYP11B2 (0.40) GRM5
SCHEMBL16800806 0.84 CYP11B2 (0.36) GRM5HSD11B1
SCHEMBL16799577 0.84 GRM5 (0.34) GRM5
SCHEMBL16800859 0.83 GRM5 (0.33) GRM5
SCHEMBL20382916 0.82 GRM5 (0.34) GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015083130-A1 FUSED PYRIDINE AND PYRIMIDINE DERIVATIVES AS ROR GAMMA MODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2015-06-11 WO disclosed
WO-2015083130-A1 FUSED PYRIDINE AND PYRIMIDINE DERIVATIVES AS ROR GAMMA MODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2015-06-11 WO disclosed