SCHEMBL16801068

SCHEMBL16801068

CC1(c2ccccc2)CCc2nc(Cl)ccc2C1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.45
HSD11B1 P28845 4/20 0.33
MEN1 O00255 1/20 0.33
CYP2C9 P11712 1/20 0.33
KMT2A Q03164 1/20 0.33
CYP11B1 P15538 1/20 0.32
CYP11B2 P19099 1/20 0.32
ALDH1A1 P00352 2/20 0.31
CYP2C19 P33261 1/20 0.31
ESR1 P03372 1/20 0.30
ESR2 Q92731 1/20 0.30
MAPT P10636 3/20 0.30
GAA P10253 1/20 0.30
RAB9A P51151 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
PLIN1 O60240 1/20 0.30
PLIN5 Q00G26 1/20 0.30
ABHD5 Q8WTS1 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
MMP1 P03956 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16798942 0.89 GRM5 (0.37) GRM5HSD11B1MEN1CYP2C9KMT2A
SCHEMBL16801056 0.87 CCR2 (0.40) GRM5HSD11B1MEN1KMT2A
SCHEMBL16800949 0.86 GRM5 (0.36) GRM5HSD11B1ALDH1A1ESR1ESR2
SCHEMBL16799547 0.86 GRM5 (0.36) GRM5HSD11B1
SCHEMBL16800950 0.85 DRD1 (0.37) GRM5ESR1ESR2
SCHEMBL16800681 0.84 MAPT (0.38) GRM5MEN1CYP2C9KMT2AALDH1A1
SCHEMBL16799325 0.84 GRM5 (0.41) GRM5MEN1KMT2A
SCHEMBL16800806 0.83 CYP11B2 (0.36) GRM5HSD11B1CYP11B1CYP11B2
SCHEMBL16799448 0.83 CYP11B2 (0.40) GRM5CYP11B1CYP11B2RAB9A
SCHEMBL16799577 0.83 GRM5 (0.34) GRM5CYP11B2ALDH1A1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015083130-A1 FUSED PYRIDINE AND PYRIMIDINE DERIVATIVES AS ROR GAMMA MODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2015-06-11 WO disclosed