SCHEMBL16800256

SCHEMBL16800256

C=CCOCCNc1ccc(CC(CNC(=O)OC(C)(C)C)CNC(=O)OC(C)(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.39
HTR1A P08908 1/20 0.39
CTSS P25774 6/20 0.36
CTSK P43235 5/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
NAMPT P43490 2/20 0.35
SYK P43405 1/20 0.35
ITGB3 P05106 1/20 0.35
ITGA2B P08514 1/20 0.35
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
ATM Q13315 1/20 0.34
MALT1 Q9UDY8 1/20 0.34
IDO1 P14902 1/20 0.34
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CTSL P07711 1/20 0.33
CTSB P07858 1/20 0.33
EGFR P00533 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18748451 0.77 SYK (0.50) CTSSCTSKSYKATMIDO1
SCHEMBL16800275 0.75
SCHEMBL13114987 0.74 TDP1 (0.47) ADRB2HTR1AL3MBTL1IDO1TDP1
SCHEMBL16800247 0.73 SYK (0.43) CTSSCTSKL3MBTL1SYKATM
SCHEMBL6874903 0.73 SYK (0.50) CTSSCTSKSYKATMIDO1
SCHEMBL23728637 0.71 ADRB2 (0.47) ADRB2HTR1AIDO1TDP1EGFR
SCHEMBL30980669 0.71 ADRB2 (0.47) ADRB2HTR1AIDO1TDP1EGFR
SCHEMBL21106804 0.71 ADRB2 (0.47) ADRB2HTR1AIDO1TDP1EGFR
SCHEMBL7408378 0.70 ATM (0.54) CTSSCTSKSYKATMIDO1
SCHEMBL21221563 0.70 LOXL2 (0.46) CTSSCTSKNAMPTSYKATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9056141-B2 Thiol-ene click chemistry for drug conjugates SYNCHEM, INC. (US) 2015-06-16 US disclosed