SCHEMBL16800677

SCHEMBL16800677

CCOC(=O)c1ccc(C2(C)CCc3nc(Cl)ccc3C2=O)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.41
NPSR1 Q6W5P4 4/20 0.41
GAA P10253 1/20 0.41
THRB P10828 2/20 0.40
TP53 P04637 1/20 0.40
MAPK1 P28482 1/20 0.38
MAPT P10636 2/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
ESR1 P03372 1/20 0.37
CA7 P43166 1/20 0.37
CA9 Q16790 1/20 0.37
ESR2 Q92731 1/20 0.37
CA14 Q9ULX7 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 4/20 0.36
LMNA P02545 2/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16800949 0.81 GRM5 (0.36) CA1CA2ESR1CA7CA9
SCHEMBL16798942 0.80 GRM5 (0.37) NPSR1MAPK1MAPTALDH1A1MAOA
SCHEMBL16799547 0.78 GRM5 (0.36) HSD17B10
SCHEMBL16800859 0.77 GRM5 (0.33)
SCHEMBL16800806 0.75 CYP11B2 (0.36)
SCHEMBL18248717 0.74 GRM5 (0.33)
SCHEMBL16800950 0.72 DRD1 (0.37) ESR1ESR2
SCHEMBL30646147 0.71 GRM5 (0.36) ESR1ESR2
SCHEMBL18248716 0.70 GRM5 (0.35) ALDH1A1LMNAKMT2ACYP2C9CYP2C19
SCHEMBL30646121 0.70 GRM5 (0.39) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015083130-A1 FUSED PYRIDINE AND PYRIMIDINE DERIVATIVES AS ROR GAMMA MODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2015-06-11 WO disclosed