SCHEMBL16801035

SCHEMBL16801035

CC1(c2ccccc2Cl)CCC(N)=CC1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 4/20 0.41
GRIN2A Q12879 4/20 0.41
SLC6A4 P31645 2/20 0.41
GRIN2D O15399 2/20 0.41
GRIN3B O60391 2/20 0.41
GRIN2B Q13224 2/20 0.41
GRIN2C Q14957 2/20 0.41
GRIN3A Q8TCU5 2/20 0.41
OPRK1 P41145 1/20 0.41
LMNA P02545 1/20 0.41
OPRM1 P35372 1/20 0.41
CACNA1C Q13936 1/20 0.41
TAAR1 Q96RJ0 1/20 0.39
HSD11B1 P28845 2/20 0.37
HDAC4 P56524 1/20 0.35
TSHR P16473 1/20 0.33
SRD5A1 P18405 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
PGR P06401 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16799589 0.72 GRIN1 (0.47) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
SCHEMBL19479822 0.70 GRIN1 (0.63) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
SCHEMBL19992375 0.70 GRIN1 (0.63) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
SCHEMBL16801016 0.69 TAAR1 (0.36) TAAR1HSD11B1
SCHEMBL16879814 0.69 GRIN1 (0.40) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
SCHEMBL16880299 0.68 ALDH1A1 (0.39) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
SCHEMBL4329065 0.67 CYP19A1 (0.32)
SCHEMBL16799023 0.65 GRIN1 (0.38) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B
SCHEMBL31668779 0.65 MAOA (0.41) LMNAHSD11B1
SCHEMBL5897472 0.65 TAAR1 (0.44) GRIN1GRIN2ASLC6A4GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015083130-A1 FUSED PYRIDINE AND PYRIMIDINE DERIVATIVES AS ROR GAMMA MODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2015-06-11 WO disclosed