SCHEMBL16801016

SCHEMBL16801016

CC1(c2ccc(Br)cc2)CCC(N)=CC1=O

nearest known ligand 0.36

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.36
CYP19A1 P11511 2/20 0.35
HSD11B1 P28845 3/20 0.34
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27040318 0.70 CYP19A1 (0.47) CYP19A1
SCHEMBL20805424 0.70 CYP19A1 (0.47) CYP19A1
SCHEMBL16800674 0.70 HSD11B1 (0.38) TAAR1CYP19A1HSD11B1HSD17B10
SCHEMBL4329065 0.69 CYP19A1 (0.32) CYP19A1
SCHEMBL16801035 0.69 GRIN1 (0.41) TAAR1HSD11B1
SCHEMBL19586055 0.64 MMP1 (0.39) CYP19A1HSD11B1
SCHEMBL4333448 0.63 TSHR (0.34) CYP19A1
SCHEMBL30912373 0.63 GRIN1 (0.42) CYP19A1HSD11B1HSD17B10
SCHEMBL28617264 0.63 KDM1A (0.42)
SCHEMBL16799247 0.63 ALDH1A1 (0.32) CYP19A1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015083130-A1 FUSED PYRIDINE AND PYRIMIDINE DERIVATIVES AS ROR GAMMA MODULATORS AURIGENE DISCOVERY TECHNOLOGIES LIMITED (IN) 2015-06-11 WO disclosed