SCHEMBL16812973

SCHEMBL16812973

O=C1CC(CO)=C(c2ccncc2)c2[nH]c3ccccc3c2N1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 5/20 0.39
CDK5R1 Q15078 5/20 0.39
CCNB2 O95067 3/20 0.39
CDK1 P06493 3/20 0.39
CCNB1 P14635 3/20 0.39
CCNB3 Q8WWL7 3/20 0.39
CCNT1 O60563 2/20 0.39
CCNA2 P20248 2/20 0.39
CDK2 P24941 2/20 0.39
CDK9 P50750 2/20 0.39
CCNA1 P78396 2/20 0.39
CCNT2 O60583 1/20 0.39
GSK3B P49841 3/20 0.38
GSK3A P49840 1/20 0.38
MAPK14 Q16539 3/20 0.37
IMPDH2 P12268 2/20 0.36
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
FNTA P49354 1/20 0.36
FNTB P49356 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16796663 0.88 CYP11B1 (0.43) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL16812964 0.86 CDK5 (0.47) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL16813043 0.83 IMPDH2 (0.46) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL16813029 0.78 CCNB2 (0.43) CCNB2CDK1CCNB1CCNB3IMPDH2
SCHEMBL16812968 0.76 CDK5 (0.46) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL16812972 0.76 GSK3B (0.46) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL16812974 0.72 SMN1; SMN2 (0.44) CDK5CDK5R1MAPK14IMPDH2PARP1
SCHEMBL16796624 0.71 CYP11B1 (0.53) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL16813039 0.69 CDK5 (0.50) CDK5CDK5R1CCNB2CDK1CCNB1
SCHEMBL16796639 0.67 MMP2 (0.43) CCNB2CDK1CCNB1CCNB3FNTA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015088565-A1 P2X4 RECEPTOR MODULATING COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC. (US) 2015-06-18 WO disclosed