SCHEMBL16824857

SCHEMBL16824857

COC[C@@]1(C(C)(C)C)CN(c2ccc([N+](=O)[O-])cc2CO)CCN1C(=O)O

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 12/20 0.40
LMNA P02545 8/20 0.40
MAPT P10636 7/20 0.40
SMN1; SMN2 Q16637 4/20 0.37
GAA P10253 3/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
KDM4E B2RXH2 1/20 0.36
KCNJ1 P48048 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16824835 0.83 MAPT (0.52) ALDH1A1LMNAMAPTSMN1; SMN2GAA
SCHEMBL16824939 0.83 MAPT (0.52) ALDH1A1LMNAMAPTSMN1; SMN2GAA
SCHEMBL1814622 0.74 ALDH1A1 (0.65) ALDH1A1LMNAMAPTSMN1; SMN2GAA
SCHEMBL30310805 0.74 ALDH1A1 (0.65) ALDH1A1LMNAMAPTSMN1; SMN2GAA
SCHEMBL16570120 0.73 LMNA (0.57) ALDH1A1LMNAMAPTSMN1; SMN2GAA
SCHEMBL17958742 0.73 LMNA (0.57) ALDH1A1LMNAMAPTSMN1; SMN2GAA
SCHEMBL1813408 0.73 MAPT (0.67) ALDH1A1LMNAMAPTSMN1; SMN2
SCHEMBL18186426 0.71 ALDH1A1 (0.60) ALDH1A1LMNAMAPTSMN1; SMN2GAA
SCHEMBL16824823 0.71 ALDH1A1 (0.60) ALDH1A1LMNAMAPTSMN1; SMN2GAA
SCHEMBL1971542 0.71 ALDH1A1 (0.57) ALDH1A1LMNASMN1; SMN2GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3083625-A1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS Almac Discovery Limited (GB) 2016-10-26 EP disclosed
WO-2015092431-A1 PYRIMIDOPYRIMIDINONES USEFUL AS WEE-1 KINASE INHIBITORS ALMAC DISCOVERY LIMITED (GB) 2015-06-25 WO disclosed