SCHEMBL16876752

SCHEMBL16876752

CC(C)(C)OC(=O)N1CCC(Nc2cc(F)c(C#N)cc2N)CC1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 10/20 0.52
NSD2 O96028 2/20 0.47
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 1/20 0.46
MAPT P10636 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
DPP4 P27487 1/20 0.43
EHMT2 Q96KQ7 1/20 0.43
EPHX1 P07099 1/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC2 Q92769 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4646790 0.89 NSD2 (0.48) GPR119NSD2ALDH1A1NPC1MAPT
SCHEMBL18425256 0.88 ALDH1A1 (0.56) GPR119ALDH1A1NPC1MAPTMAPK1
SCHEMBL3107643 0.85 ALDH1A1 (0.50) GPR119ALDH1A1NPC1MAPTMAPK1
SCHEMBL28331009 0.84 GPR119 (0.37) GPR119NSD2
SCHEMBL16876736 0.84 L3MBTL1 (0.50) GPR119NSD2ALDH1A1NPC1MAPT
SCHEMBL15410448 0.84 ALDH1A1 (0.49) GPR119NSD2ALDH1A1NPC1MAPT
SCHEMBL4647276 0.83 ALDH1A1 (0.50) GPR119NSD2ALDH1A1NPC1MAPT
SCHEMBL4434545 0.82 ALDH1A1 (0.50) GPR119NSD2ALDH1A1NPC1MAPT
SCHEMBL4648718 0.82 ALDH1A1 (0.49) GPR119NSD2ALDH1A1NPC1MAPT
SCHEMBL4647099 0.82 ALDH1A1 (0.51) GPR119ALDH1A1NPC1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3092228-A1 TRPA1 MODULATORS Algomedix, Inc. (US) 2016-11-16 EP disclosed
WO-2015103060-A1 TRPA1 MODULATORS ALGOMEDIX, INC. (US) 2015-07-09 WO disclosed