SCHEMBL16888281

SCHEMBL16888281

CCn1cc2c(n1)CCC(C)(C)C2

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.35
HTT P42858 3/20 0.34
GAA P10253 1/20 0.33
HDAC9 Q9UKV0 3/20 0.33
PDK1 Q15118 1/20 0.32
MAPK1 P28482 1/20 0.32
KMT2A Q03164 1/20 0.32
HTR2C P28335 1/20 0.31
TSHR P16473 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19132763 0.84 RORC (0.36) RORCHTTGAAHDAC9KMT2A
SCHEMBL19132768 0.80 HTT (0.60) HTTGAAKMT2ATSHRSMN1; SMN2
SCHEMBL19132769 0.78 HTT (0.43) HTTGAAHDAC9MAPK1KMT2A
SCHEMBL19132756 0.77 PDK1 (0.34) RORCPDK1MAPK1HTR2C
SCHEMBL18217031 0.75 RORC (0.33) RORCHDAC9KMT2A
SCHEMBL18896278 0.73 HTT (0.59) HTTGAAKMT2ATSHRSMN1; SMN2
SCHEMBL17682605 0.73 HTT (0.54) HTTGAAKMT2ATSHRSMN1; SMN2
SCHEMBL12507439 0.69 SMN1; SMN2 (0.31) HTTSMN1; SMN2
SCHEMBL12489633 0.68 HTR2C (0.48) HTTGAAKMT2AHTR2CSMN1; SMN2
SCHEMBL12691665 0.68 CYP2C19 (0.41) HTTGAAKMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015103507-A1 CYCLOHEXYL SULFONE RORϒ MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2015-07-09 WO disclosed