SCHEMBL1688901

SCHEMBL1688901

O=c1c2cn(C3CCOCC3)nc2nc(-c2ccccc2F)n1-c1ccc(Br)cc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.42
ALDH1A2 O94788 7/20 0.42
ALDH1A3 P47895 7/20 0.42
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CNR1 P21554 2/20 0.35
CNR2 P34972 2/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
PDE1A P54750 1/20 0.35
PDE1B Q01064 1/20 0.35
PDE1C Q14123 1/20 0.35
TRPV4 Q9HBA0 1/20 0.34
TP53 P04637 1/20 0.34
TDO2 P48775 1/20 0.32
IDO2 Q6ZQW0 1/20 0.32
GRM1 Q13255 1/20 0.32
KDM4E B2RXH2 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1688983 0.92 ALDH1A1 (0.40) ALDH1A1ALDH1A2ALDH1A3MEN1KMT2A
SCHEMBL5612554 0.89 ALDH1A1 (0.38) ALDH1A1ALDH1A2ALDH1A3MEN1KMT2A
SCHEMBL5611589 0.81 ALDH1A1 (0.45) ALDH1A1ALDH1A2ALDH1A3MEN1KMT2A
SCHEMBL1753242 0.80 PDE1C (0.55) MAPTPDE1APDE1BPDE1CTP53
SCHEMBL5611595 0.78 GRM1 (0.41) ALDH1A1ALDH1A2ALDH1A3MEN1KMT2A
SCHEMBL1688938 0.77 MEN1 (0.39) ALDH1A1ALDH1A2ALDH1A3MEN1KMT2A
SCHEMBL12088143 0.76 CNR1 (0.39) CNR1CNR2PDE1APDE1BPDE1C
SCHEMBL1688895 0.76 ALDH1A1 (0.43) ALDH1A1ALDH1A2ALDH1A3MEN1KMT2A
SCHEMBL5611874 0.75 ADORA3 (0.41) ALDH1A1MEN1KMT2AMAPTHTT
SCHEMBL1688909 0.75 ALDH1A1 (0.41) ALDH1A1ALDH1A2ALDH1A3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807429-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM, LLC (BM) 2007-07-18 EP claimed
WO-2006047516-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2006-05-04 WO claimed