SCHEMBL1689135

SCHEMBL1689135

O=c1[nH]c(-c2ccc(-c3cccc(F)c3)cc2)nc2c1nc(-c1ccc(Cl)cc1)n2-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 6/20 0.49
ALDH1A1 P00352 2/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.47
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
BLM P54132 1/20 0.45
PLEC Q15149 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
DHODH Q02127 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
TNKS O95271 3/20 0.41
TNKS2 Q9H2K2 3/20 0.41
PARP2 Q9UGN5 2/20 0.41
GUSB P08236 1/20 0.41
RXFP1 Q9HBX9 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39
PARP1 P09874 1/20 0.39
MAPK13 O15264 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5611669 0.92 DHFR (0.51) DHFRALDH1A1HPGDTSHRLMNA
SCHEMBL5611463 0.86 DHFR (0.64) DHFRALDH1A1TSHRLMNAHTT
SCHEMBL1689302 0.84 DHFR (0.49) DHFRALDH1A1HPGDTSHRLMNA
SCHEMBL5611470 0.83 DHFR (0.55) DHFRALDH1A1HPGDTSHRLMNA
SCHEMBL5611734 0.83 DHFR (0.55) DHFRALDH1A1HPGDTSHRLMNA
SCHEMBL5611607 0.81 DHFR (0.47) DHFRALDH1A1HPGDTSHRKDM4E
SCHEMBL5611495 0.81 DHFR (0.50) DHFRALDH1A1HPGDTSHRLMNA
SCHEMBL5611826 0.80 DHFR (0.49) DHFRALDH1A1HPGDTSHRLMNA
SCHEMBL5612502 0.80 DHFR (0.53) DHFRALDH1A1HPGDTSHRTNKS
SCHEMBL4750784 0.80 DHFR (0.53) DHFRALDH1A1HPGDTSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1807429-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM, LLC (BM) 2007-07-18 EP claimed
WO-2006047516-A2 COMPOUNDS AND COMPOSITIONS AS INHIBITORS OF CANNABINOID RECEPTOR 1 ACTIVITY IRM LLC (BM) 2006-05-04 WO claimed