SCHEMBL16896807

SCHEMBL16896807

CC(C(N)=O)c1c(F)cccc1S(C)(=O)=O

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
GBA1 P04062 1/20 0.35
KAT6A Q92794 2/20 0.35
SLC9A1 P19634 2/20 0.34
APP P05067 1/20 0.34
SLC9A2 Q9UBY0 1/20 0.34
PTGS2 P35354 1/20 0.33
LOX P28300 1/20 0.33
HTT P42858 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2C P18825 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33
ADRA1B P35368 1/20 0.33
CNR2 P34972 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29718627 0.83 CES2 (0.46) CES2CES1APP
SCHEMBL24603708 0.80 CNR2 (0.37) CES2CES1GBA1KAT6AADRA2A
SCHEMBL16896758 0.73 MMP2 (0.45) SLC9A1SLC9A2LOX
SCHEMBL14938633 0.72 APP (0.52) APPPTGS2
SCHEMBL19717529 0.71 CES2 (0.39) CES2CES1SLC9A1HTT
SCHEMBL11076456 0.69 CYP1A2 (0.37) SLC9A1SLC9A2LOX
SCHEMBL2061390 0.69 ADRA2A (0.38) ADRA2AADRA2CADRA1DADRA1AADRA1B
SCHEMBL2642086 0.69 ALB (0.44) CES2CES1PTGS2HTTADRA2A
SCHEMBL8491731 0.68 CES2 (0.47) CES2CES1KAT6APTGS2HTT
SCHEMBL775432 0.68 PTGES2 (0.46) CES2CES1KAT6APTGS2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3091970-A1 LXR AGONISTS AND USES THEREOF Rgenix, Inc. (US) 2016-11-16 EP disclosed
WO-2015106164-A1 LXR AGONISTS AND USES THEREOF RGENIX, INC. (US) 2015-07-16 WO disclosed