Predicted protein targets (top 19)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | LMNA | P02545 | 2/20 | 0.50 |
| ▸ | EHMT2 | Q96KQ7 | 1/20 | 0.46 |
| ▸ | EHMT1 | Q9H9B1 | 1/20 | 0.46 |
| ▸ | APOBEC3G | Q9HC16 | 1/20 | 0.46 |
| ▸ | ALDH1A1 | P00352 | 7/20 | 0.44 |
| ▸ | SMN1; SMN2 | Q16637 | 4/20 | 0.42 |
| ▸ | KMT2A | Q03164 | 2/20 | 0.41 |
| ▸ | MAPT | P10636 | 2/20 | 0.41 |
| ▸ | RAB9A | P51151 | 5/20 | 0.40 |
| ▸ | HPGD | P15428 | 3/20 | 0.40 |
| ▸ | NPC1 | O15118 | 2/20 | 0.40 |
| ▸ | KDM4E | B2RXH2 | 1/20 | 0.40 |
| ▸ | ALOX15 | P16050 | 1/20 | 0.40 |
| ▸ | HSD17B10 | Q99714 | 1/20 | 0.40 |
| ▸ | PKM | P14618 | 2/20 | 0.38 |
| ▸ | MEN1 | O00255 | 1/20 | 0.38 |
| ▸ | POLB | P06746 | 2/20 | 0.38 |
| ▸ | MAPK10 | P53779 | 1/20 | 0.37 |
| ▸ | RGS12 | O14924 | 1/20 | 0.37 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL25399704 | 0.92 | LMNA (0.48) | LMNAEHMT2EHMT1APOBEC3GALDH1A1 | |
| SCHEMBL29573871 | 0.89 | LMNA (0.46) | LMNAEHMT2EHMT1APOBEC3GALDH1A1 | |
| SCHEMBL1425231 | 0.88 | LMNA (0.52) | LMNAEHMT2EHMT1APOBEC3GALDH1A1 | |
| SCHEMBL28254695 | 0.85 | LMNA (0.52) | LMNAEHMT2EHMT1APOBEC3GALDH1A1 | |
| SCHEMBL28494764 | 0.79 | LMNA (0.57) | LMNAEHMT2EHMT1APOBEC3GALDH1A1 | |
| Butyric Acid SCHEMBL15845048 | 0.78 | ALDH1A1 (0.61) | LMNAEHMT2EHMT1APOBEC3GALDH1A1 | |
| SCHEMBL535803 | 0.77 | LMNA (0.50) | LMNAEHMT2EHMT1APOBEC3GALDH1A1 | |
| SCHEMBL29224770 | 0.75 | LMNA (0.43) | LMNAEHMT2EHMT1APOBEC3GALDH1A1 | |
| SCHEMBL12893090 | 0.75 | LMNA (0.48) | LMNAEHMT2EHMT1APOBEC3GALDH1A1 | |
| SCHEMBL28529987 | 0.75 | EHMT2 (0.47) | LMNAEHMT2EHMT1APOBEC3GALDH1A1 |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| CN-113769108-B | Conjugates of cysteine engineered antibodies | 伊缪诺金公司 | 2024-11-08 | — | — | CN | disclosed |
| EP-4366777-A2 | LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME | PROFOUNDBIO US CO. (US) | 2024-05-15 | — | — | EP | disclosed |
| WO-2023160376-A1 | ANTIBODIES AND VARIANTS THEREOF AGAINST HUMAN B7-H3 | NANJING PROBIO BIOTECH CO., LTD. (CN) | 2023-08-31 | — | — | WO | disclosed |
| CN-115850449-A | Antibodies and conjugates | 苏州智核生物医药科技有限公司 | 2023-03-28 | — | — | CN | disclosed |
| EP-4149546-A1 | DRUG CONJUGATES CONTAINING ALPHA-ENOLASE ANTIBODIES AND USES THEREOF | Hunilife Biotechnology, Inc. (TW) | 2023-03-22 | — | — | EP | disclosed |
| WO-2023280227-A2 | LINKERS, DRUG LINKERS AND CONJUGATES THEREOF AND METHODS OF USING THE SAME | PROFOUNDBIO US CO. (US) | 2023-01-12 | — | — | WO | disclosed |
| WO-2021228044-A1 | DRUG CONJUGATES CONTAINING ALPHA-ENOLASE ANTIBODIES AND USES THEREOF | HUNILIFE BIOTECHNOLOGY, INC. (CN) | 2021-11-18 | — | — | WO | disclosed |
| EP-3189082-A1 | ANTI-PD-L1 CONJUGATES FOR TREATING TUMORS | Birdie Biopharmaceuticals Inc. (KY) | 2017-07-12 | — | — | EP | disclosed |
| EP-3092254-A1 | COMPOUNDS AND COMPOSITIONS FOR TREATING HER2 POSITIVE TUMORS | Birdie Biopharmaceuticals Inc. (KY) | 2016-11-16 | — | — | EP | disclosed |
| EP-3092255-A1 | COMPOUNDS AND COMPOSITIONS FOR TREATING EGFR EXPRESSING TUMORS | Birdie Biopharmaceuticals Inc. (KY) | 2016-11-16 | — | — | EP | disclosed |
| EP-3092256-A1 | COMPOUNDS AND COMPOSITIONS FOR IMMUNOTHERAPY | Shanghai Birdie Biotech Inc. (CN) | 2016-11-16 | — | — | EP | disclosed |
| WO-2016034085-A1 | ANTI-PD-L1 CONJUGATES FOR TREATING TUMORS | BIRDIE BIOPHARMACEUTICALS, INC. (KY) | 2016-03-10 | — | — | WO | disclosed |
| WO-2015103987-A1 | COMPOUNDS AND COMPOSITIONS FOR TREATING HER2 POSITIVE TUMORS | SHANGHAI BIRDIE BIOTECH, INC. (CN) | 2015-07-16 | — | — | WO | disclosed |
| WO-2015103989-A1 | COMPOUNDS AND COMPOSITIONS FOR IMMUNOTHERAPY | SHANGHAI BIRDIE BIOTECH, INC. (CN) | 2015-07-16 | — | — | WO | disclosed |
| WO-2015103990-A1 | COMPOUNDS AND COMPOSITIONS FOR TREATING EGFR EXPRESSING TUMORS | SHANGHAI BIRDIE BIOTECH, INC. (CN) | 2015-07-16 | — | — | WO | disclosed |