SCHEMBL16909354

SCHEMBL16909354

COC(=O)C1(NC(=O)OC(C)(C)C)CCN(c2ncc(B(O)O)cn2)CC1

nearest known ligand 0.36

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.36
GPR119 Q8TDV5 7/20 0.34
RET P07949 8/20 0.34
MAPT P10636 1/20 0.33
PPIA P62937 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15539980 0.90 GPR119 (0.34) CYP3A4GPR119RETMAPT
SCHEMBL21639716 0.87 CYP3A4 (0.37) CYP3A4GPR119RETMAPTPPIA
SCHEMBL1282700 0.87 CYP3A4 (0.37) CYP3A4GPR119RETMAPTPPIA
SCHEMBL28719905 0.86 RET (0.42) RET
SCHEMBL20137774 0.85 RET (0.43) CYP3A4GPR119RETMAPT
SCHEMBL15416347 0.83 CYP3A4 (0.40) CYP3A4GPR119RETPPIA
SCHEMBL15415397 0.78 CYP3A4 (0.42) CYP3A4MAPT
SCHEMBL15415493 0.78 CYP3A4 (0.42) CYP3A4RETMAPT
SCHEMBL16909548 0.77 CYP3A4 (0.44) CYP3A4MAPT
SCHEMBL1282440 0.76 PANK3 (0.39) CYP3A4GPR119RETMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2872508-B1 IMIDAZOPYRIDINE DERIVATIVES AS MODULATORS OF TNF ACTIVITY UCB BIOPHARMA SPRL (BE) 2018-08-29 EP disclosed
US-9309243-B2 Imidazopyridine derivatives as modulators of TNF activity UCB BIOPHARMA SPRL (BE) 2016-04-12 US disclosed
US-20150203486-A1 Imidazopyridine Derivatives as Modulators of TNF Activity UCB Biopharma SPRL a corporation 2015-07-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150203486-A1 Imidazopyridine Derivatives as Modulators of TNF Activity TNF, TNFRSF1A, IL1A CYP3A4 1261/4885GPR119 498/4885RET 1583/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.