SCHEMBL1691920

SCHEMBL1691920

OCCCc1c(-c2ccc(Cl)cc2)nc2ccccn12

nearest known ligand 0.63

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.63
NPC1 O15118 2/20 0.63
RAB9A P51151 2/20 0.63
POLB P06746 1/20 0.63
HTT P42858 1/20 0.63
SMN1; SMN2 Q16637 1/20 0.63
GAA P10253 1/20 0.57
SLC2A1 P11166 1/20 0.57
GABRA1 P14867 1/20 0.55
GABRA5 P31644 1/20 0.55
GABRB2 P47870 1/20 0.55
KCNK3 O14649 9/20 0.51
KCNK9 Q9NPC2 9/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1691661 0.86 KDM4E (0.69) KDM4ENPC1RAB9APOLBHTT
SCHEMBL7222018 0.85 GABRA1 (0.59) KDM4ENPC1RAB9APOLBHTT
Hydrochloric Acid SCHEMBL1430093 0.81 KDM4E (0.69) KDM4ENPC1RAB9APOLBHTT
SCHEMBL1431043 0.81 KDM4E (0.69) KDM4ENPC1RAB9APOLBHTT
SCHEMBL13341899 0.80 NPC1 (0.55) KDM4ENPC1RAB9APOLBHTT
SCHEMBL8208 0.80 KDM4E (0.64) KDM4ENPC1RAB9APOLBHTT
SCHEMBL7223975 0.79 KDM4E (0.65) KDM4ENPC1RAB9APOLBHTT
SCHEMBL7228643 0.78 KDM4E (0.64) KDM4ENPC1RAB9APOLBHTT
SCHEMBL7231135 0.78 KDM4E (0.58) KDM4ENPC1RAB9APOLBHTT
SCHEMBL1430221 0.77 KDM4E (0.67) KDM4ENPC1RAB9APOLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2376490-B1 IMIDAZOPYRIDINE COMPOUNDS PROXIMAGEN LTD (GB) 2013-01-23 EP claimed
US-20120010188-A1 Imidazopyridine Compounds PROMIMAGEN LTD. (GB) 2012-01-12 US claimed
EP-2376490-A1 IMIDAZOPYRIDINE COMPOUNDS Proximagen Limited (GB) 2011-10-19 EP claimed
WO-2010064020-A1 IMIDAZOPYRIDINE COMPOUNDS PROXIMAGEN LTD. (GB) 2010-06-10 WO claimed
US-20150239905-A1 IMIDAZOPYRIDINE COMPOUNDS BIOVITRUM AB (PUBL) (SE) 2015-08-27 US disclosed
US-20140206662-A1 Imidazopyridine Compounds PROXIMAGEN LTD. (GB) 2014-07-24 US disclosed
EP-2376490-B1 IMIDAZOPYRIDINE COMPOUNDS PROXIMAGEN LTD (GB) 2013-01-23 EP disclosed
US-20120010188-A1 Imidazopyridine Compounds PROMIMAGEN LTD. (GB) 2012-01-12 US disclosed
EP-2376490-A1 IMIDAZOPYRIDINE COMPOUNDS Proximagen Limited (GB) 2011-10-19 EP disclosed
WO-2010064020-A1 IMIDAZOPYRIDINE COMPOUNDS PROXIMAGEN LTD. (GB) 2010-06-10 WO disclosed
US-6514969-B2 Alzheimer's diseas, Parkinson disease, Huntington disease BOEHRINGER INGELHEIM PHARMA KG (DE) 2003-02-04 US disclosed
US-20020042420-A1 Beta-amyloid inhibitors, processes for preparing them, and their use in pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2002-04-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120010188-A1 Imidazopyridine Compounds SSB, MIF, IDO1 KDM4E 2671/4885NPC1 1153/4885RAB9A 3798/4885
US-20150239905-A1 IMIDAZOPYRIDINE COMPOUNDS SSB, MIF, IDO1 KDM4E 2671/4885NPC1 1153/4885RAB9A 3798/4885
US-20020042420-A1 Beta-amyloid inhibitors, processes for preparing them, and their use in pharmaceutical compositions HTT, APP, BACE1 KDM4E 4232/4885NPC1 44/4885RAB9A 2085/4885
US-20140206662-A1 Imidazopyridine Compounds SSB, NFKBIA, TPMT KDM4E 2821/4885NPC1 2286/4885RAB9A 3886/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.