SCHEMBL8208

SCHEMBL8208

O=C(O)Cc1c(-c2ccc(Cl)cc2)nc2ccccn12

nearest known ligand 0.67

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.64
NPC1 O15118 1/20 0.64
POLB P06746 1/20 0.64
HTT P42858 1/20 0.64
RAB9A P51151 1/20 0.64
SMN1; SMN2 Q16637 1/20 0.64
GABRA1 P14867 1/20 0.61
GABRA5 P31644 1/20 0.61
GABRB2 P47870 1/20 0.61
GAA P10253 1/20 0.58
SLC2A1 P11166 1/20 0.58
KCNK3 O14649 7/20 0.57
KCNK9 Q9NPC2 7/20 0.57
SLC2A2 P11168 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6686729 0.90 NTRK1 (0.58) KDM4ENPC1RAB9ASMN1; SMN2GAA
SCHEMBL7222018 0.86 GABRA1 (0.59) KDM4ENPC1POLBHTTRAB9A
SCHEMBL8150 0.85 GABRA2 (0.70) GABRB2SLC2A1SLC2A2
SCHEMBL1431027 0.85 KDM4E (0.59) KDM4ENPC1POLBHTTRAB9A
SCHEMBL1691661 0.85 KDM4E (0.69) KDM4ENPC1POLBHTTRAB9A
SCHEMBL1430614 0.83 SLC2A2 (0.77) KDM4ENPC1POLBHTTRAB9A
SCHEMBL1431043 0.82 KDM4E (0.69) KDM4ENPC1POLBHTTRAB9A
Hydrochloric Acid SCHEMBL1430093 0.82 KDM4E (0.69) KDM4ENPC1POLBHTTRAB9A
SCHEMBL13341895 0.82 NPC1 (0.56) KDM4ENPC1POLBHTTRAB9A
SCHEMBL28391511 0.81 GABRA2 (0.48) GABRB2SLC2A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060084806-A1 Processes for the preparation of imidazo[1,2-a] pyridine derivatives GLENMARK PHARMACEUTICALS LIMITED (IN) 2006-04-20 US disclosed
US-4460592-A HYPNOTIC SYNTHELABO 1984-07-17 US disclosed
US-4382938-A HYPNOSIS; TENSION; ANTICONVULSANTS; PSYCHOLOGICAL AND NERVOUS SYSTEM DISORDERS SYNTHELABO (FR) 1983-05-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060084806-A1 Processes for the preparation of imidazo[1,2-a] pyridine derivatives CBR1, HNRNPA2B1, HNRNPR KDM4E 3801/4885NPC1 1312/4885POLB 1694/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.