Triamcinolone Acetonide

Triamcinolone Acetonide

SCHEMBL1692059

CC1(C)O[C@@H]2C[C@H]3[C@@H]4CCC5=CC(=O)C=C[C@]5(C)[C@@]4(F)[C@@H](O)C[C@]3(C)[C@]2(C(=O)CO)O1.CC1(C)O[C@@H]2C[C@H]3[C@@H]4CCC5=CC(=O)C=C[C@]5(C)[C@@]4(F)[C@@H](O)C[C@]3(C)[C@]2(C(=O)CO)O1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

NR3C1

The experimentally established mechanism targets of Triamcinolone Acetonide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 known ✓ P04150 4/20 1.00
HIF1A Q16665 9/20 1.00
CYP3A4 P08684 8/20 1.00
LMNA P02545 7/20 1.00
PGR P06401 4/20 1.00
NR1I2 O75469 1/20 1.00
NPSR1 Q6W5P4 2/20 0.79
HSD17B10 Q99714 5/20 0.73
MAPT P10636 2/20 0.73
TDP1 Q9NUW8 1/20 0.73
KDM4E B2RXH2 1/20 0.73
AR P10275 1/20 0.73
MAPK1 P28482 1/20 0.73
CNR1 P21554 1/20 0.70
KCNH2 Q12809 1/20 0.70
USP2 O75604 1/20 0.70
CYP2C9 P11712 2/20 0.68
NFKB1 P19838 2/20 0.68
CYP2J2 P51589 1/20 0.68
BLM P54132 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Triamcinolone Acetonide SCHEMBL4448 1.00 HIF1A (1.00) HIF1ACYP3A4LMNANR3C1PGR
Triamcinolone Acetonide SCHEMBL16393966 1.00 HIF1A (1.00) HIF1ACYP3A4LMNANR3C1PGR
Triamcinolone Acetonide SCHEMBL4002585 1.00 HIF1A (1.00) HIF1ACYP3A4LMNANR3C1PGR
Triamcinolone Acetonide SCHEMBL12323208 1.00 HIF1A (1.00) HIF1ACYP3A4LMNANR3C1PGR
Triamcinolone Acetonide SCHEMBL5484214 1.00 HIF1A (1.00) HIF1ACYP3A4LMNANR3C1PGR
Triamcinolone Acetonide SCHEMBL13234864 1.00 HIF1A (1.00) HIF1ACYP3A4LMNANR3C1PGR
Triamcinolone Acetonide SCHEMBL13839748 1.00 HIF1A (1.00) HIF1ACYP3A4LMNANR3C1PGR
Triamcinolone Acetonide SCHEMBL11332717 1.00 HIF1A (1.00) HIF1ACYP3A4LMNANR3C1PGR
Triamcinolone Acetonide SCHEMBL21051778 1.00 HIF1A (1.00) HIF1ACYP3A4LMNANR3C1PGR
Triamcinolone Acetonide SCHEMBL11911289 1.00 HIF1A (1.00) HIF1ACYP3A4LMNANR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 66 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220177574-A1 FcgammaRIIB-Specific Antibodies and Methods of Use Thereof MACROGENICS, INC. (US) 2022-06-09 US disclosed
US-20200131265-A1 FcgammaRIIB-Specific Antibodies and Methods of Use Thereof MACROGENICS, INC. (US) 2020-04-30 US disclosed
US-10584181-B2 Methods of making and using multispecific antibody panels and antibody analog panels GENENTECH, INC. (US) 2020-03-10 US disclosed
US-20190218288-A1 FcgammaRIIB-Specific Antibodies and Methods of Use Thereof MACROGENICS, INC. (US) 2019-07-18 US disclosed
US-10100116-B2 FcγRIIB-specific antibodies and methods of use thereof MACROGENICS, INC. (US) 2018-10-16 US disclosed
EP-2029173-B1 FC RIIB-SPECIFIC ANTIBODIES AND METHODS OF USE THEREOF MACROGENICS INC (US) 2016-07-20 EP disclosed
EP-1534335-B9 FCGAMMARIIB-SPECIFIC ANTIBODIES AND METHODS OF USE THEREOF MACROGENICS INC (US) 2016-01-13 EP disclosed
US-20150344574-A1 FcGammaRIIB Specific Antibodies and Methods of Use Thereof MACROGENICS, INC. (US) 2015-12-03 US disclosed
US-20150344575-A1 FcGammaRIIB Specific Antibodies and Methods of Use Thereof MACROGENICS, INC. (US) 2015-12-03 US disclosed
US-9084799-B2 Inhaled combination therapy PULMAGEN THERAPEUTICS (SYNERGY) LIMITED (GB) 2015-07-21 US disclosed
US-20060013810-A1 Humanized FcgammaRIIB-specific antibodies and methods of use thereof MACROGENICS, INC. 2006-01-19 US disclosed
WO-2005115452-A2 FCϜRIIB-SPECIFIC ANTIBODIES AND METHODS OF USE THEREOF MACROGENICS, INC. (US) 2005-12-08 WO disclosed
US-20050260213-A1 Fcgamma-RIIB-specific antibodies and methods of use thereof MACROGENICS, INC. 2005-11-24 US disclosed
WO-2005110474-A2 HUMANIZED FcϜRIIB SPECIFIC ANTIBODIES AND METHODS OF USE THEREOF MACROGENICS, INC. (US) 2005-11-24 WO disclosed
US-20050215767-A1 Fcgamma riib specific antibodies and methods of use thereof MACROGENICS INC. 2005-09-29 US disclosed
EP-1534335-A2 FCGAMMARIIB-SPECIFIC ANTIBODIES AND METHODS OF USE THEREOF MACROGENICS, INC. (US) 2005-06-01 EP disclosed
WO-2005018669-A1 FCϜRIIB-SPECIFIC ANTIBODIES AND METHODS OF USE THEREOF MACROGENICS, INC. (US) 2005-03-03 WO disclosed
US-20040185045-A1 FcgammaRIIB-specific antibodies and methods of use thereof MACROGENICS, INC. 2004-09-23 US disclosed
WO-2004016750-A2 FcϜRIIB-SPECIFIC ANTIBODIES AND METHODS OF USE THEREOF MACROGENICS, INC. (US) 2004-02-26 WO disclosed
US-4920180-A Hydrophilic polymer MENICON CO., LTD. (JP) 1990-04-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10584181-B2 Methods of making and using multispecific antibody panels and antibody analog panels FCGR2A, FCGR3B, FCGR1A NR3C1 1811/4885HIF1A 4674/4885CYP3A4 1650/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.