SCHEMBL16935293

SCHEMBL16935293

CCOc1[nH]c(=O)c(C#N)c2c1CCCC2

nearest known ligand 0.61

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.61
KDM4E B2RXH2 6/20 0.61
HPGD P15428 6/20 0.61
KMT2A Q03164 1/20 0.61
HSD11B1 P28845 12/20 0.58
CYP1A2 P05177 1/20 0.56
CYP2D6 P10635 1/20 0.56
CYP2C9 P11712 1/20 0.56
HIF1A Q16665 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29740984 0.76 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDKMT2AHSD11B1
SCHEMBL7271706 0.74 ALDH1A1 (1.00) ALDH1A1KDM4EHPGDKMT2AHSD11B1
SCHEMBL16935203 0.72 ALDH1A1 (0.96) ALDH1A1KDM4EHPGDKMT2AHSD11B1
SCHEMBL24256907 0.71 ALDH1A1 (0.94) ALDH1A1KDM4EHPGDKMT2AHSD11B1
SCHEMBL9846227 0.70 ALDH1A1 (0.93) ALDH1A1KDM4EHPGDKMT2AHSD11B1
SCHEMBL15923482 0.70 ALDH1A1 (0.63) ALDH1A1KDM4EHPGDKMT2AHSD11B1
SCHEMBL16935255 0.68 ALDH1A1 (0.60) ALDH1A1KDM4EHPGDKMT2AHSD11B1
SCHEMBL14499342 0.67 POLB (0.76) ALDH1A1KDM4EHPGDKMT2ACYP1A2
SCHEMBL16935340 0.67 ALDH1A1 (0.58) ALDH1A1KDM4EHPGDKMT2AHSD11B1
SCHEMBL16935353 0.65 ALDH1A1 (0.56) ALDH1A1KDM4EHPGDKMT2AHSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015110999-A1 EZH2 INHIBITORS AND USES THEREOF Piramal Enterprises Limited (IN) 2015-07-30 WO disclosed