SCHEMBL1695138

SCHEMBL1695138

N#C[C@H](O)c1ccccc1[N+](=O)[O-]

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
ALDH1A1 P00352 7/20 0.49
TSHR P16473 2/20 0.47
MAPT P10636 2/20 0.47
CDK5 Q00535 1/20 0.47
CDK5R1 Q15078 1/20 0.47
HPGD P15428 1/20 0.46
GPR35 Q9HC97 1/20 0.42
PLAU P00749 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
HSD17B10 Q99714 1/20 0.41
SGMS2 Q8NHU3 1/20 0.40
TDP1 Q9NUW8 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1694369 1.00 CYP1A2 (0.50) CYP1A2ALDH1A1TSHRMAPTCDK5
SCHEMBL1695140 1.00 CYP1A2 (0.50) CYP1A2ALDH1A1TSHRMAPTCDK5
SCHEMBL28374691 0.82 CYP1A2 (0.50) CYP1A2ALDH1A1TSHRMAPTCDK5
SCHEMBL3697952 0.81 CYP1A2 (0.59) CYP1A2ALDH1A1TSHRGPR35PLAU
SCHEMBL13937393 0.80 TSHR (0.61) ALDH1A1TSHRMAPTMEN1KMT2A
SCHEMBL8136284 0.80 GPR35 (0.48) ALDH1A1TSHRMAPTCDK5CDK5R1
SCHEMBL28414312 0.79 ALDH1A1 (0.50) CYP1A2ALDH1A1TSHRMAPTCDK5
SCHEMBL31014201 0.79 CYP1A2 (0.58) CYP1A2ALDH1A1TSHRGPR35PLAU
SCHEMBL8521008 0.79 CYP1A2 (0.58) CYP1A2ALDH1A1TSHRGPR35PLAU
SCHEMBL506668 0.79 CYP1A2 (0.58) CYP1A2ALDH1A1TSHRGPR35PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8969573-B2 Compounds for the inhibition of cellular proliferation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2015-03-03 US disclosed
US-20130178505-A1 Compounds for the Inhibition of Cellular Proliferation PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2013-07-11 US disclosed
EP-2585453-A2 COMPOUNDS FOR THE INHIBITION OF CELLULAR PROLIFERATION President and Fellows of Harvard College (US) 2013-05-01 EP disclosed
WO-2012006068-A2 COMPOUNDS FOR THE INHIBITION OF CELLULAR PROLIFERATION PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2012-01-12 WO disclosed
CN-100445375-C Modified nitrilases and their use in methods for the production of carboxylic acids BASF AG (DE) 2008-12-24 CN disclosed
CN-1753990-A Modified nitrilases and their use in methods for the production of carboxylic acids BASF AG (DE) 2006-03-29 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130178505-A1 Compounds for the Inhibition of Cellular Proliferation MKI67, EIF2AK2, CDK2 CYP1A2 4741/4885ALDH1A1 3428/4885TSHR 4098/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.