SCHEMBL16972798

SCHEMBL16972798

O=c1cc(CCc2cccc(O)c2)oc2cc(O)ccc12

nearest known ligand 0.77

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2B P41595 3/20 0.67
LOXL2 Q9Y4K0 1/20 0.59
PPARG P37231 2/20 0.57
MEN1 O00255 1/20 0.55
TNKS O95271 1/20 0.55
ALDH1A1 P00352 1/20 0.55
CYP3A4 P08684 1/20 0.55
PARP1 P09874 1/20 0.55
CYP2C9 P11712 1/20 0.55
HPGD P15428 1/20 0.55
KMT2A Q03164 1/20 0.55
TNKS2 Q9H2K2 1/20 0.55
HTR3A P46098 1/20 0.52
AKR1B1 P15121 3/20 0.51
HSD17B3 P37058 2/20 0.51
CA12 O43570 1/20 0.49
AKR1B10 O60218 1/20 0.49
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CYP1A2 P05177 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16972788 0.90 PPARG (0.71) HTR2BLOXL2PPARGHTR3AAKR1B1
SCHEMBL16972870 0.89 PPARG (0.74) HTR2BPPARGMEN1TNKSCYP3A4
SCHEMBL16972770 0.87 LOXL2 (0.64) HTR2BLOXL2PPARGALDH1A1CYP3A4
SCHEMBL18417922 0.81 HTR2B (1.00) HTR2BCYP3A4HTR3A
SCHEMBL16972796 0.80 LOXL2 (0.58) HTR2BLOXL2PPARGMEN1HPGD
SCHEMBL29129664 0.79 PPARG (0.70) HTR2BLOXL2PPARGMEN1TNKS
SCHEMBL27806527 0.79 PPARG (0.71) HTR2BPPARGALDH1A1CYP3A4HPGD
SCHEMBL30335890 0.79 PPARG (0.71) HTR2BPPARGALDH1A1CYP3A4HPGD
SCHEMBL7901121 0.77 LOXL2 (0.71) LOXL2MEN1TNKSALDH1A1CYP3A4
SCHEMBL3661429 0.77 ALOX15 (0.72) LOXL2PPARGALDH1A1CYP3A4HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015116460-A1 2-SUBSTITUTED-5-HYDROXY-4H-CHROMEN-4-ONES AS NOVEL LIGANDS FOR THE SEROTONIN RECEPTOR 2B (5-HT2B) VIRGINIA COMMONWEALTH UNIVERSITY (US) 2015-08-06 WO claimed