SCHEMBL16984239

SCHEMBL16984239

CCc1c(-c2ccc(N3CCC(N(C)C)C3)cc2)[nH]c(=O)c2c(=O)[nH]n(C)c12

nearest known ligand 0.68

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.68
MCHR1 Q99705 10/20 0.39
TLR9 Q9NR96 3/20 0.37
TLR7 Q9NYK1 3/20 0.37
TLR8 Q9NR97 2/20 0.37
SYK P43405 1/20 0.37
PDGFRB P09619 1/20 0.36
FGFR1 P11362 1/20 0.36
KDR P35968 1/20 0.36
RORC P51449 2/20 0.34
FLT3 P36888 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16972734 0.82 KCNH2 (0.60) KCNH2MCHR1TLR9TLR7TLR8
SCHEMBL16972703 0.81 KCNH2 (1.00) KCNH2MCHR1TLR9TLR7TLR8
SCHEMBL14758924 0.77 KCNH2 (0.62) KCNH2MCHR1TLR9TLR7TLR8
Hydrochloric Acid SCHEMBL14745204 0.76 KCNH2 (0.61) KCNH2MCHR1TLR9TLR7TLR8
SCHEMBL16972737 0.74 KCNH2 (0.59) KCNH2MCHR1TLR9TLR7TLR8
SCHEMBL16567839 0.74 KCNH2 (0.61) KCNH2MCHR1SYKPDGFRBFGFR1
SCHEMBL14758835 0.73 KCNH2 (0.57) KCNH2MCHR1PDGFRBFGFR1KDR
SCHEMBL14758820 0.73 KCNH2 (0.57) KCNH2MCHR1PDGFRBFGFR1KDR
SCHEMBL14745687 0.73 KCNH2 (0.57) KCNH2MCHR1PDGFRBFGFR1KDR
Hydrochloric Acid SCHEMBL14745362 0.72 KCNH2 (0.56) KCNH2MCHR1PDGFRBFGFR1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015114317-A1 5H-ISOTHIAZOLO[4,5-C]PYRIDINE-3,4-DIONE OR 5H-PYRAZOLO[4,3-C]PYRIDIN-3,4-DIONE AS ANTIBACTERIAL COMPOUNDS REDX PHARMA PLC (GB) 2015-08-06 WO disclosed