SCHEMBL1699205

SCHEMBL1699205

Cc1cnc2c([nH]c(=O)n2-c2ccc(O)cc2)c1C(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
MAP3K11 Q16584 6/20 0.40
KDM4E B2RXH2 3/20 0.39
GAA P10253 3/20 0.39
HSD17B10 Q99714 2/20 0.39
MAPK1 P28482 1/20 0.39
MTOR P42345 2/20 0.36
HPGD P15428 2/20 0.36
USP2 O75604 1/20 0.36
ESR1 P03372 2/20 0.35
ESR2 Q92731 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34
MAPK14 Q16539 1/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699227 0.84 MEN1 (0.44) MEN1KMT2AMAP3K11KDM4EGAA
SCHEMBL1699234 0.81 L3MBTL1 (0.54) PIK3CACSNK2A1
SCHEMBL1699264 0.80 MAP3K11 (0.40) MEN1KMT2AMAP3K11KDM4EGAA
SCHEMBL15385957 0.78 MAP3K11 (0.41) MEN1KMT2AMAP3K11KDM4EGAA
SCHEMBL1699212 0.76 MAP3K11 (0.40) MEN1KMT2AMAP3K11KDM4EGAA
SCHEMBL1699111 0.73 PDE10A (0.36) MEN1KMT2AHSD17B10USP2MAPK13
SCHEMBL1699627 0.72 KDM4E (0.40) MEN1KMT2AMAP3K11KDM4EGAA
SCHEMBL1699169 0.72 MAP3K11 (0.39) MEN1KMT2AMAP3K11KDM4EGAA
SCHEMBL1699077 0.70 MAP3K11 (0.39) MEN1KMT2AMAP3K11KDM4EGAA
SCHEMBL1699349 0.70 MAP3K11 (0.38) MEN1KMT2AMAP3K11KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed