SCHEMBL1699210

SCHEMBL1699210

CCc1ccnc2c1[nH]c(=O)n2-c1ccc(Oc2nc3cccnc3[nH]2)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD1 P21728 4/20 0.38
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.36
PABPC1 P11940 1/20 0.36
PKM P14618 1/20 0.35
TP53 P04637 1/20 0.35
KDM4C Q9H3R0 3/20 0.34
PDE4B Q07343 1/20 0.34
MET P08581 3/20 0.34
TSHR P16473 1/20 0.33
PDGFRB P09619 1/20 0.33
KIT P10721 1/20 0.33
PDGFRA P16234 1/20 0.33
FLT4 P35916 1/20 0.33
KDR P35968 1/20 0.33
FLT3 P36888 1/20 0.33
ALK Q9UM73 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699363 0.84 KDM4C (0.39) KDM4C
SCHEMBL9981014 0.78 ADORA3 (0.38) DRD1MEN1KMT2APOLBPABPC1
SCHEMBL14889112 0.77 DRD1 (0.38) DRD1ALDH1A1MEN1KMT2APOLB
SCHEMBL12045529 0.75 LTA4H (0.43) ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL1701784 0.74 LTA4H (0.42) ALDH1A1MEN1KMT2A
SCHEMBL9981008 0.74 LTA4H (0.41) MEN1KMT2A
SCHEMBL1699182 0.74 NPC1 (0.37) ALDH1A1MEN1KMT2APKMTSHR
SCHEMBL9981668 0.73 GABRP (0.51)
SCHEMBL1699077 0.73 MAP3K11 (0.39) ALDH1A1MEN1KMT2ATSHR
SCHEMBL1699098 0.72 DRD1 (0.44) DRD1MEN1KMT2APOLBPABPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed