SCHEMBL16992168

SCHEMBL16992168

Cn1nnnc1C1CCN(C(=O)O)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.34
ALDH1A1 P00352 5/20 0.34
HTR2B P41595 1/20 0.34
GAA P10253 2/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.32
CACNA1C Q13936 1/20 0.32
TSHR P16473 1/20 0.32
KDM4E B2RXH2 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
USP2 O75604 1/20 0.32
ALOX15 P16050 1/20 0.32
MAPK1 P28482 1/20 0.32
CASP1 P29466 1/20 0.32
CASP7 P55210 1/20 0.32
HSD17B10 Q99714 1/20 0.32
DPP4 P27487 1/20 0.31
GPR4 P46093 1/20 0.31
HPGD P15428 1/20 0.30
PRCP P42785 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16992432 0.79 HSD11B1 (0.38) ALDH1A1LMNAMAPTUSP2DPP4
SCHEMBL31076314 0.79 NPC1 (0.36) ALDH1A1GAALMNATSHRKDM4E
SCHEMBL15017310 0.76 SMN1; SMN2 (0.57) SMN1; SMN2
SCHEMBL3170060 0.76 TRPV1 (0.39) EPHX2ALDH1A1GAALMNAMAPT
SCHEMBL21774900 0.75 GAA (0.42) ALDH1A1GAAHPGD
SCHEMBL21774899 0.75 GAA (0.42) ALDH1A1GAAHPGD
SCHEMBL2391972 0.75 HPGDS (0.44) ALDH1A1MAPTKDM4EHPGD
SCHEMBL2391975 0.75 HPGDS (0.44) ALDH1A1MAPTKDM4EHPGD
SCHEMBL9933978 0.74 ALDH1A1 (0.31) ALDH1A1GAALMNA
SCHEMBL9940153 0.74 ALDH1A1 (0.31) ALDH1A1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3102568-A1 BICYCLIC AZA COMPOUNDS AS MUSCARINIC M1 RECEPTOR AND/OR M4 RECEPTOR AGONISTS Heptares Therapeutics Limited (GB) 2016-12-14 EP disclosed
WO-2015118342-A1 BICYCLIC AZA COMPOUNDS AS MUSCARINIC M1 RECEPTOR AGONISTS. HEPTARES THERAPEUTICS LIMITED (GB) 2015-08-13 WO disclosed