SCHEMBL1699268

SCHEMBL1699268

O=c1[nH]c2cc(OCC(F)(F)F)cnc2n1CCc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.43
PLAT P00750 1/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C9 P11712 2/20 0.41
TSHR P16473 2/20 0.41
CYP2C19 P33261 2/20 0.41
CYP2D6 P10635 1/20 0.41
HRH3 Q9Y5N1 3/20 0.40
HMOX1 P09601 2/20 0.40
PDE2A O00408 1/20 0.39
CTSV O60911 1/20 0.38
CTSL P07711 1/20 0.38
FFAR1 O14842 2/20 0.38
FFAR4 Q5NUL3 2/20 0.38
FAAH O00519 1/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4C Q9H3R0 1/20 0.38
LMNA P02545 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699530 0.84 CYP1A2 (0.45) MAOBPLATALDH1A1CYP1A2CYP2C9
SCHEMBL14889030 0.73 HRH3 (0.42) MAOBHRH3HMOX1PDE2AFFAR1
SCHEMBL4340540 0.71 LMNA (0.60) MAOBCYP1A2CYP2C19LMNAHIF1A
SCHEMBL1699299 0.70 NPC1 (0.45) MAOBNPC1RAB9AL3MBTL1
SCHEMBL1699357 0.69 PRMT5 (0.50) ALDH1A1CYP1A2CYP2C9TSHRCYP2C19
SCHEMBL9981622 0.68 NPC1 (0.58) MAOBALDH1A1CTSVCTSLMEN1
SCHEMBL1699176 0.66 NPC1 (0.49) MAOBCTSVCTSLMEN1KMT2A
SCHEMBL1699265 0.65 NPC1 (0.46) MAOBALDH1A1TSHRMEN1KMT2A
SCHEMBL24861854 0.64 MAOB (0.62) MAOB
SCHEMBL29192686 0.64 MAOB (0.76) MAOBCTSVCTSLMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed