SCHEMBL1699357

SCHEMBL1699357

Cc1ccnc2c1[nH]c(=O)n2CCc1ccc(OCc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT5 O14744 2/20 0.50
HMOX1 P09601 1/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
HRH3 Q9Y5N1 3/20 0.44
PKM P14618 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
ALDH1A1 P00352 3/20 0.43
CYP1A2 P05177 2/20 0.43
CYP2C9 P11712 2/20 0.43
TSHR P16473 2/20 0.43
CYP2C19 P33261 2/20 0.43
LMNA P02545 1/20 0.43
CYP3A4 P08684 1/20 0.43
HIF1A Q16665 1/20 0.43
CYP2D6 P10635 1/20 0.43
F2 P00734 1/20 0.42
KCNH2 Q12809 1/20 0.42
GRIN2B Q13224 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699310 0.82 NPC1 (0.59) PRMT5NPC1RAB9AL3MBTL1PKM
SCHEMBL1699530 0.74 CYP1A2 (0.45) HMOX1NPC1RAB9AL3MBTL1HRH3
SCHEMBL1699268 0.69 MAOB (0.43) HMOX1NPC1RAB9AL3MBTL1HRH3
SCHEMBL28068238 0.69 ADORA3 (0.57) NPC1RAB9AL3MBTL1SMN1; SMN2ALDH1A1
SCHEMBL1699548 0.69 NPC1 (0.59) PRMT5NPC1RAB9AL3MBTL1PKM
SCHEMBL8713816 0.67 ADORA2B (0.50) TSHRKMT2AMEN1ADORA3ADORA2B
SCHEMBL1699470 0.67 NPC1 (0.54) PRMT5NPC1RAB9AL3MBTL1PKM
SCHEMBL1699315 0.67 NPC1 (0.50) PRMT5NPC1RAB9AL3MBTL1PKM
SCHEMBL9126862 0.67 AGTR2 (0.63)
SCHEMBL21951965 0.66 ALDH1A1 (0.56) ALDH1A1LMNAKMT2AHPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed