SCHEMBL1699284

SCHEMBL1699284

O=c1[nH]c2c(C3CC3)ccnc2n1-c1ccc(O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K11 Q16584 7/20 0.39
HPGD P15428 1/20 0.38
LMNA P02545 1/20 0.36
ESR1 P03372 1/20 0.36
ESR2 Q92731 1/20 0.36
MTOR P42345 1/20 0.34
CCNE1 P24864 3/20 0.33
CDK2 P24941 3/20 0.33
PIK3CD O00329 2/20 0.33
PIK3CA P42336 2/20 0.33
PIK3CB P42338 2/20 0.33
PIK3CG P48736 2/20 0.33
CCNT1 O60563 1/20 0.33
CDK1 P06493 1/20 0.33
CDK4 P11802 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNA2 P20248 1/20 0.33
CCND1 P24385 1/20 0.33
CDK9 P50750 1/20 0.33
CCNE2 O96020 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15385957 0.79 MAP3K11 (0.41) MAP3K11HPGDLMNAESR1ESR2
SCHEMBL1699077 0.76 MAP3K11 (0.39) MAP3K11HPGDLMNAESR1ESR2
SCHEMBL1699133 0.70 DAO (0.58) MAP3K11ESR1ESR2ALDH1A1
SCHEMBL1702888 0.69 MAP3K11 (0.36) MAP3K11HPGDLMNAESR1ESR2
SCHEMBL1699227 0.67 MEN1 (0.44) MAP3K11HPGDESR1ESR2MTOR
SCHEMBL1699212 0.67 MAP3K11 (0.40) MAP3K11HPGDLMNAESR1ESR2
SCHEMBL1699205 0.66 MEN1 (0.43) MAP3K11HPGDESR1ESR2MTOR
SCHEMBL1699264 0.66 MAP3K11 (0.40) MAP3K11HPGDLMNAESR1ESR2
SCHEMBL1699169 0.65 MAP3K11 (0.39) MAP3K11HPGDLMNAESR1ESR2
SCHEMBL1699627 0.65 KDM4E (0.40) MAP3K11HPGDLMNAESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed