SCHEMBL1699291

SCHEMBL1699291

CCc1cnc2c([nH]c(=O)n2-c2ccccc2O)c1C

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.40
BRD4 O60885 1/20 0.38
GAA P10253 4/20 0.36
MAPK13 O15264 3/20 0.36
MAPK12 P53778 3/20 0.36
MAPK11 Q15759 3/20 0.36
MAPK14 Q16539 3/20 0.36
KDM4E B2RXH2 2/20 0.36
POLB P06746 2/20 0.36
ALDH1A1 P00352 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
HPGD P15428 2/20 0.36
GLA P06280 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
DAO P14920 1/20 0.35
NPEPPS P55786 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
HIF1A Q16665 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1699212 0.80 MAP3K11 (0.40) HSP90AA1GAAKDM4EALDH1A1HPGD
SCHEMBL10790345 0.66 BRD4 (0.56) HSP90AA1BRD4GAAKDM4EPOLB
SCHEMBL9120324 0.66 AURKA (0.58) HSP90AA1BRD4GAAKDM4EPOLB
SCHEMBL1699349 0.64 MAP3K11 (0.38) GAAKDM4EALDH1A1HPGDDAO
SCHEMBL1699264 0.64 MAP3K11 (0.40) GAAMAPK13MAPK12MAPK11MAPK14
SCHEMBL1699169 0.61 MAP3K11 (0.39) GAAMAPK13MAPK12MAPK11MAPK14
SCHEMBL9119078 0.61 HSP90AA1 (0.72) HSP90AA1BRD4GAAKDM4EPOLB
SCHEMBL10027225 0.61 LMNA (0.43) GAAKDM4EPOLBALDH1A1HPGD
SCHEMBL8544900 0.59 POLB (0.65) BRD4GAAKDM4EPOLBALDH1A1
SCHEMBL15385957 0.58 MAP3K11 (0.41) GAAMAPK13MAPK12MAPK11MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed