SCHEMBL16994909

SCHEMBL16994909

CC(=O)[C@@H](NC(=O)[C@@H]1CCCN1C(=O)Cc1ccc(-c2ccccc2)cc1)[C@@H](C)O

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.52
MME P08473 1/20 0.48
MMEL1 Q495T6 1/20 0.48
ITGB1 P05556 5/20 0.46
ITGA4 P13612 5/20 0.46
VHL P40337 1/20 0.46
ACE P12821 3/20 0.46
CPA1 P15085 1/20 0.44
CPA2 P48052 1/20 0.44
CPA4 Q9UI42 1/20 0.44
ELANE P08246 1/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
PKM P14618 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL403446 0.91 SLC6A2 (0.50) SLC6A2MMEMMEL1ITGB1ITGA4
SCHEMBL6543907 0.79 CPA1 (0.51) ITGB1ITGA4ACECPA1CPA2
SCHEMBL5037359 0.79 GYS1 (0.56) MMEMMEL1ACE
SCHEMBL5037364 0.79 GYS1 (0.56) MMEMMEL1ACE
SCHEMBL6353403 0.78 ACE (0.50) ACEELANE
SCHEMBL20707067 0.78 CYP3A4 (0.52) ITGB1ITGA4ACECYP3A4CYP2C9
SCHEMBL6354335 0.76 PSMB9 (0.51) ITGB1ITGA4
SCHEMBL14723759 0.76 ALDH1A1 (0.59) ITGB1ITGA4CYP2C9CYP2C19
SCHEMBL10956149 0.76 F2 (0.48) ITGB1ITGA4ACECPA1CPA2
SCHEMBL5040451 0.75 GYS1 (0.52) MMEMMEL1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295402-B1 Antibacterial agents UNIV WASHINGTON (US) 2015-08-12 EP disclosed