SCHEMBL1701343

SCHEMBL1701343

CC(C)(C)c1cc(Oc2nc3ccccc3n2COCC[Si](C)(C)C)ccc1OC(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.41
F2R P25116 1/20 0.36
KDM4E B2RXH2 5/20 0.36
HSD17B10 Q99714 3/20 0.36
RECQL P46063 1/20 0.36
CYP2C9 P11712 1/20 0.35
ALDH1A1 P00352 4/20 0.35
TP53 P04637 2/20 0.35
HPGD P15428 1/20 0.35
MAPK1 P28482 1/20 0.35
RAB9A P51151 1/20 0.35
PIN1 Q13526 2/20 0.35
KCNH2 Q12809 1/20 0.35
CNR2 P34972 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
PTGDR2 Q9Y5Y4 1/20 0.34
TSHR P16473 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9980956 0.76 KDM4E (0.44) NPC1KDM4EHSD17B10ALDH1A1TP53
SCHEMBL23123437 0.76 SMN1; SMN2 (0.45) NPC1KDM4EHSD17B10ALDH1A1TP53
SCHEMBL1701488 0.75 PIN1 (0.38) NPC1KDM4EHSD17B10ALDH1A1TP53
SCHEMBL1701344 0.74 BRD4 (0.44) NPC1KDM4EALDH1A1TP53HPGD
SCHEMBL9981197 0.74 F11 (0.43) NPC1KDM4EALDH1A1TP53RAB9A
SCHEMBL14889062 0.72 KDM4E (0.39) NPC1KDM4EHSD17B10ALDH1A1TP53
SCHEMBL4321671 0.68 GPR119 (0.47)
SCHEMBL4577155 0.68 GPR119 (0.47)
SCHEMBL5953265 0.67 KDM4E (0.55) NPC1KDM4EHSD17B10RECQLALDH1A1
SCHEMBL23122597 0.67 NPC1 (0.39) NPC1KDM4EHSD17B10ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011163355-A1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-12-29 WO disclosed