SCHEMBL1701865

SCHEMBL1701865

Cc1c(-c2cccs2)n[nH]c1-c1ccc(N)nc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FYN P06241 1/20 0.43
MAPT P10636 3/20 0.42
PDGFRB P09619 2/20 0.39
KIT P10721 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ALPL P05186 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
POLB P06746 1/20 0.39
KDR P35968 1/20 0.39
ADK P55263 3/20 0.38
GPR119 Q8TDV5 1/20 0.38
TP53 P04637 1/20 0.37
CDK5 Q00535 1/20 0.36
CDK5R1 Q15078 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
CCNE2 O96020 2/20 0.36
CDK4 P11802 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2591881 0.85 MAPT (0.45) MAPTPDGFRBKITKDM4EALDH1A1
SCHEMBL2827765 0.77 FYN (0.56) FYNPDGFRBKDM4EALDH1A1HSD17B10
SCHEMBL1701229 0.76 PDPK1 (0.40) FYNMAPTPDGFRBKITKDM4E
SCHEMBL624711 0.75 MEN1 (0.45) MAPTKDM4EALDH1A1ALPLHPGD
SCHEMBL8684518 0.70 ILK (0.50) MAPTKDM4EALDH1A1HSD17B10POLB
SCHEMBL5499265 0.67 CYP3A4 (0.52) FYNMAPTPDGFRBKDM4EALDH1A1
SCHEMBL14088054 0.66 CYP2C9 (0.55) MAPTPDGFRBKDM4EALDH1A1HPGD
Hydrochloric Acid SCHEMBL15312178 0.65 PDGFRB (0.70) PDGFRBKITKDRCDK2CHEK1
SCHEMBL5210609 0.65 SMN1; SMN2 (0.49) MAPTKDM4EALDH1A1ALPLHPGD
SCHEMBL1701249 0.65 KDM4E (0.41) MAPTKDM4EALDH1A1ALPLHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563776-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2013-03-06 EP disclosed
WO-2011139489-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA INC. (US) 2011-11-10 WO disclosed