SCHEMBL17025751

SCHEMBL17025751

CCC(N(NC(=O)c1cc(OC)c(C)c(OC)c1)C(=O)c1ccc2c(c1C)OCCO2)C(C)(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.41
NPC1 O15118 8/20 0.38
RAB9A P51151 7/20 0.38
SMN1; SMN2 Q16637 7/20 0.38
MAPT P10636 5/20 0.38
GAA P10253 1/20 0.38
CASP1 P29466 1/20 0.38
TP53 P04637 5/20 0.38
TSHR P16473 3/20 0.38
ALDH1A1 P00352 4/20 0.37
RXFP1 Q9HBX9 2/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
MAPK1 P28482 1/20 0.36
APOBEC3A P31941 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
CREBBP Q92793 1/20 0.35
TAS2R8 Q9NYW2 1/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17416637 0.94 PLK1 (0.39) PLK1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL29684822 0.93 PLK1 (0.39) PLK1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL667456 0.93 PLK1 (0.39) PLK1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL18091873 0.89 NPC1 (0.39) NPC1RAB9ASMN1; SMN2MAPTTP53
SCHEMBL667482 0.87 PLK1 (0.37) PLK1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL29684841 0.87 PLK1 (0.37) PLK1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL667440 0.87 PLK1 (0.37) PLK1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL29684483 0.87 PLK1 (0.37) PLK1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL9903268 0.83 ALDH1A1 (0.38) NPC1RAB9ASMN1; SMN2MAPTALDH1A1
SCHEMBL29685124 0.81 ABCB1 (0.38) NPC1RAB9ASMN1; SMN2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20150240244-A1 BIOAVAILABLE DIACYLHYDRAZINE LIGANDS FOR MODULATING THE EXPRESSION OF EXOGENOUS GENES VIA AN ECDYSONE RECEPTOR COMPLEX BIOPHARMA CREDIT PLC, AS COLLATERAL AGENT (GB) 2015-08-27 US claimed