SCHEMBL17027156

SCHEMBL17027156

FC(F)(F)c1ccc2c(CBr)c[nH]c2c1

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 1/20 0.56
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP1A2 P05177 1/20 0.49
HPGD P15428 1/20 0.49
ALOX12 P18054 1/20 0.49
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.49
CDK2 P24941 3/20 0.46
DYRK1A Q13627 2/20 0.45
GPR84 Q9NQS5 2/20 0.45
GSK3B P49841 1/20 0.44
KIF11 P52732 6/20 0.44
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12327114 0.83 TBXAS1 (0.56) TBXAS1MEN1ALDH1A1CYP1A2HPGD
SCHEMBL3184412 0.83 TBXAS1 (0.52) TBXAS1MEN1ALDH1A1CYP1A2HPGD
SCHEMBL27220751 0.81 HTR2A (0.59) TBXAS1ALDH1A1CYP1A2HTR2A
SCHEMBL27220749 0.81 HTR2A (0.59) TBXAS1ALDH1A1CYP1A2HTR2A
SCHEMBL2537034 0.81 HTR2A (0.65) TBXAS1MEN1CYP1A2KMT2AHTR2A
SCHEMBL13715393 0.81 TBXAS1 (0.53) TBXAS1MEN1ALDH1A1CYP1A2HPGD
SCHEMBL6029337 0.80 CSNK2A1 (0.53) TBXAS1MEN1ALDH1A1CYP1A2HPGD
SCHEMBL6031020 0.80 MEN1 (0.55) TBXAS1MEN1ALDH1A1CYP1A2HPGD
SCHEMBL2386812 0.78 ALDH1A1 (0.58) TBXAS1MEN1ALDH1A1CYP1A2HPGD
SCHEMBL6031147 0.77 ICMT (0.63) TBXAS1MEN1ALDH1A1CYP1A2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107910-A1 NEW PHENYLAZETIDINE, CARBOXYLATE OR CARBOXAMIDE COMPOUNDS INVENTIVA (FR) 2016-12-28 EP disclosed
WO-2015124868-A1 NEW PHENYLAZETIDINE, CARBOXYLATE OR CARBOXAMIDE COMPOUNDS INVENTIVA (FR) 2015-08-27 WO disclosed